Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263692 (US9714221, Example 29) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263669 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263674 (US9714221, Example 11) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263673 (6-(2-fluoro- 4-hydroxy- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263691 (6- (benzofuran- 5-yl)-5- [4-[(3S)-1- (3- fluoropro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263686 (6-(2- chloro-4- methyl- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263892 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263719 (6-(1,3- benzoxazol- 5-yl)-5-[4- [(3S)-1-(3- fluoro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263712 (6-(2,3- dihydro- 1,4- benzodioxin-6-yl)-5- [4-[(3S...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263690 (6-(4- ethoxy-2- methyl- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263677 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263755 (6-(2- chloro-4- methoxy- phenyl)-5- [4-[(3S)-1- (3...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263671 (6-(2- chloro-3- fluoro- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263693 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263683 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263672 (US9714221, Example 36 | US9714221, Example 9) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263675 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263697 (6-(6- ethoxy-3- pyridyl)-5- [4-[(3S)-1- (3- fluoro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263706 (6-(2- chloro-4- ethoxy- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263893 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263676 (6-(4- chloro-3- methyl- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263694 (6-(2,3- dimethyl- phenyl)-5-[4- [(3S)-1-(3- fluoro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263707 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263764 (6-(2,2- dimethyl- 3H- benzo- furan-5-yl)-5- [4-[(3...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263743 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 13 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263847 (6-(2,2-dimethylindolin-5-yl)-5-[4-[(3S)-1-(3-fluor...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263680 (6-(4-fluoro- 2-methyl- phenyl)-5- [4-[(3S)-1- (3- ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 15 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263900 (6-[2,3- difluoro-4- (1-piperidyl)- phenyl]-5- [4-[...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 15 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263860 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263748 (US9714221, Example 82) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263709 (6-(4- ethoxy-2- methyl- phenyl)-1- fluoro-5-[4- [(...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263770 (6-(2-fluoro- 6-methoxy- 3-pyridyl)- 5-[4-[(3S)- 1-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263775 (US9714221, Example 109) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263757 (5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263737 (6-(6- ethoxy-2- fluoro-3- pyridyl)-5- [4-[(3S)- 1-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263670 (6-(3- chloro-2- methyl- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263911 (US9714221, Example 207) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263774 (US9714221, Example 108) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263843 (6-(6- ethoxy-5- fluoro-3- pyridyl)-5- [4-[(3S)-1- ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263681 (6-(2,4- dichloro- phenyl)-5-[4- [(3S)-1-(3- fluoro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 21 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263668 (6-(2- chloro-4- fluoro- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 21 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263736 (US9714221, Example 70) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 22 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263665 (5-[4-[(3S)- 1-(3- fluoro- propyl)pyrrolidin- 3-yl]...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 22 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263664 (US9714221, Example 1) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 22 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263708 (US9714221, Example 45) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263742 (US9714221, Example 76) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263917 (6-(2-chloro-4-fluoro-phenyl)-1-fluoro-5-[4-[(3S)-1...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263710 (6-(2,4- dichloro- phenyl)-1- fluoro-5-[4- [(3S)-1-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263788 (6-(2- chloro-3- fluoro- phenyl)-1- fluoro-5-[4- [(...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 24 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Estrogen receptor [Y537S] (Homo sapiens (Human)) | BDBM263678 (6-(4- chloro-2- fluoro- phenyl)-5- [4-[(3S)-1- (3-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 24 | n/a | n/a | n/a | n/a | 7.4 | 25 |
SANOFI US Patent | Assay Description It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b... | US Patent US9714221 (2017) BindingDB Entry DOI: 10.7270/Q2N58PB1 | |||||||||||
More data for this Ligand-Target Pair |
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