Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM24183 (4-amino-n-[2,3-3H]butyric acid | 4-aminobutanoic a...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50020883 ((R)-Piperidine-3-carboxylic acid | (R)-nipecotic a...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039246 ((S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piper...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.09E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ludwig-Maximilians-University Munich Curated by ChEMBL | Assay Description Inhibition of rat GAT2 assessed as [3H]GABA uptake | Bioorg Med Chem 19: 6492-504 (2011) Article DOI: 10.1016/j.bmc.2011.08.039 BindingDB Entry DOI: 10.7270/Q2154JB8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039234 (1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-pipe...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.ejmech.2022.114269 BindingDB Entry DOI: 10.7270/Q2JM2FM0 | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039246 ((S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piper...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039245 (CHEMBL309357 | Dimethyl-[2-(1,7,7-trimethyl-2-phen...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents | PubMed | n/a | n/a | 3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039234 (1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-pipe...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039242 (1-{2-[Bis-(4-chloro-phenyl)-(4-methoxy-phenyl)-met...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50003624 ((RS)-nipecotic acid | CHEMBL277498 | Nipecotic | P...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 3.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039235 (1-{2-[(4-Methoxy-phenyl)-di-p-tolyl-methoxy]-ethyl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039238 (1-{2-[Bis-(4-fluoro-phenyl)-(4-methoxy-phenyl)-met...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039233 (1-{2-[9-(4-Methoxy-phenyl)-9H-fluoren-9-yloxy]-eth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ludwig-Maximilians-University Munich Curated by ChEMBL | Assay Description Inhibition of rat GAT2-mediated GABA uptake | Eur J Med Chem 46: 1483-98 (2011) Article DOI: 10.1016/j.ejmech.2011.01.042 BindingDB Entry DOI: 10.7270/Q2F76CWJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039233 (1-{2-[9-(4-Methoxy-phenyl)-9H-fluoren-9-yloxy]-eth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039233 (1-{2-[9-(4-Methoxy-phenyl)-9H-fluoren-9-yloxy]-eth...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Ludwig-Maximilians-Universit£t M£nchen Curated by ChEMBL | Assay Description Inhibition of rat GAT-2 expressed in thymidine kinase deficient mouse LM cells assessed as decrease in [3H]GABA uptake after 10 mins by scintillation... | Eur J Med Chem 124: 852-880 (2016) Article DOI: 10.1016/j.ejmech.2016.09.012 BindingDB Entry DOI: 10.7270/Q27M09XT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM90787 (1,2,3,6-tetrahydropyridine-5-carboxylic acid;hydro...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039240 (1-{2-[Bis-(4-methoxy-phenyl)-phenyl-methoxy]-ethyl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039236 (1-{2-[Tris-(4-methoxy-phenyl)-methylsulfanyl]-ethy...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039244 (1-(2-Tritylsulfanyl-ethyl)-piperidine-3-carboxylic...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 8.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039237 (1-{3-[Tris-(4-methoxy-phenyl)-methoxy]-propyl}-pip...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.03E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039249 (1-{2-[(4-Methoxy-phenyl)-diphenyl-methoxy]-ethyl}-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.37E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039241 (1-{2-[(4-Methoxy-3-trifluoromethyl-phenyl)-phenyl-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 1.77E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039248 ((R)-1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.40E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039252 (1-{2-[(3-Fluoro-4-methoxy-phenyl)-(3-fluoro-phenyl...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.17E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50403565 (CHEMBL2093978) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 4.47E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporte | Bioorg Med Chem Lett 6: 1535-1540 (1996) Article DOI: 10.1016/S0960-894X(96)00268-5 BindingDB Entry DOI: 10.7270/Q2NV9J79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50003634 (1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article | n/a | n/a | 5.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporte | Bioorg Med Chem Lett 6: 1535-1540 (1996) Article DOI: 10.1016/S0960-894X(96)00268-5 BindingDB Entry DOI: 10.7270/Q2NV9J79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50020891 ((R)-1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carbo...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50403566 (CHEMBL2094022) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 6.69E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporte | Bioorg Med Chem Lett 6: 1535-1540 (1996) Article DOI: 10.1016/S0960-894X(96)00268-5 BindingDB Entry DOI: 10.7270/Q2NV9J79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50403563 (CHEMBL2093977) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 7.57E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporte | Bioorg Med Chem Lett 6: 1535-1540 (1996) Article DOI: 10.1016/S0960-894X(96)00268-5 BindingDB Entry DOI: 10.7270/Q2NV9J79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50020888 ((S)-Piperidine-3-carboxylic acid | (S)-nipecotic a...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 7.63E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50403564 (CHEMBL2094024) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 8.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was tested for its ability to inhibit uptake of [3H]- GABA by cloned rat GAT-2 transporte | Bioorg Med Chem Lett 6: 1535-1540 (1996) Article DOI: 10.1016/S0960-894X(96)00268-5 BindingDB Entry DOI: 10.7270/Q2NV9J79 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50003618 (1-{2-[Bis-(4-trifluoromethyl-phenyl)-methoxy]-ethy...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.28E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039251 ((R)-1-(4,4-bis(3-methylthiophen-2-yl)but-3-enyl)pi...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 1.41E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039247 (1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-1,2,...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 2.80E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium- and chloride-dependent GABA transporter 2 (Rattus norvegicus) | BDBM50039253 (1-{2-[Tris-(4-fluoro-phenyl)-methoxy]-ethyl}-piper...) | KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.67E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Synaptic Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibitory activity against rat GABA transporter-2 (rGAT2) | J Med Chem 37: 2334-42 (1994) BindingDB Entry DOI: 10.7270/Q2P849XX | |||||||||||
More data for this Ligand-Target Pair |