Found 592 hits of ic50 for UniProtKB: Q92993 Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kcal/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653650
(US11911372, Example 72)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)-c1ccn[nH]1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet 
| UniChem
| US Patent
| n/a | n/a | 106 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653602
(US11911372, Example 23)Show SMILES CCc1ccc(OC)cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653593
(US11911372, Example 14)Show SMILES COc1ccc(OC(C)C)c(c1)-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 142 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653585
(US11911372, Example 6)Show SMILES COc1ccc(OC)c(c1)-c1cc(NS(=O)(=O)c2c(OC)cc(cc2OC)-c2ccccc2)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 164 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM646444
(US11911372, Example 1 | US11911372, Example 69 | U...)Show SMILES COc1ccc(Br)cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 213 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653595
(US11911372, Example 16)Show SMILES CCOc1ccc(OC)cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 219 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653688
(US11911372, Example 111)Show SMILES COc1cccc(OC)c1S(=O)(=O)Nc1nnc(s1)-c1cc(Cl)ccc1OC(C)C | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 238 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653594
(US11911372, Example 15)Show SMILES COc1ccc(Cl)cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 315 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653649
(US11911372, Example 71)Show SMILES COCc1ccc(OC)cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 416 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653587
(US11911372, Example 8)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)C1CC1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 416 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653597
(US11911372, Example 18)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)-c1ncco1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 445 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653586
(US11911372, Example 7)Show SMILES COc1ccc(OC)c(c1)-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 586 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653648
(US11911372, Example 70)Show SMILES COc1ccc(OC)c(c1)-c1nnc(NS(=O)(=O)c2c(OC)cccc2OC)s1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 696 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653696
(US11911372, Example 119)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)-c1ccnn1C | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 788 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM646444
(US11911372, Example 1 | US11911372, Example 69 | U...)Show SMILES COc1ccc(Br)cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 845 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653590
(US11911372, Example 11)Show SMILES COc1ccccc1-c1cc(NS(=O)(=O)c2c(OC)cc(cc2OC)-c2ccccc2)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 867 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653584
(US11911372, Example 5)Show SMILES CCOc1ccccc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653682
(US11911372, Example 105)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)-n1cccn1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653651
(US11911372, Example 73)Show SMILES COCc1ccc(OC)c(c1)-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 1.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653601
(US11911372, Example 22)Show SMILES COc1cccc(OC)c1S(=O)(=O)Nc1cc(on1)-c1ccccc1OC(F)(F)F | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 1.34E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653697
(US11911372, Example 120)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)-c1cn[nH]c1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 1.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653634
(US11911372, Example 56)Show SMILES COc1ccccc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 1.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653662
(US11911372, Example 84)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)-c1ccccc1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 1.84E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM50151660
(CHEMBL3774630)Show InChI InChI=1S/C6H4N2S4/c1-3-7-9-5(1)11-12-6-2-4-8-10-6/h1-4H | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
MCE
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Freiburg
Curated by ChEMBL
| Assay Description
Inhibition of recombinant N-terminal His-tagged TIP60 (unknown origin) expressed in baculovirus-infected insect cell system using histone substrate i... |
J Med Chem 59: 1249-70 (2016)
Article DOI: 10.1021/acs.jmedchem.5b01502
BindingDB Entry DOI: 10.7270/Q2DV1MRN |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM50151660
(CHEMBL3774630)Show InChI InChI=1S/C6H4N2S4/c1-3-7-9-5(1)11-12-6-2-4-8-10-6/h1-4H | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
MCE
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sichuan University
Curated by ChEMBL
| Assay Description
Inhibition of Tip60 (unknown origin) using [3H]-acetyl-CoA as substrate preincubated for 10 mins followed by substrate addition measured after 10 min... |
Eur J Med Chem 178: 259-286 (2019)
Article DOI: 10.1016/j.ejmech.2019.05.078
BindingDB Entry DOI: 10.7270/Q2ZW1QC8 |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM50151660
(CHEMBL3774630)Show InChI InChI=1S/C6H4N2S4/c1-3-7-9-5(1)11-12-6-2-4-8-10-6/h1-4H | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
MCE
KEGG
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sichuan University
Curated by ChEMBL
| Assay Description
Displacement of [3H]-acetyl-CoA from recombinant Tip60 (unknown origin) by scintillation counting analysis |
Eur J Med Chem 178: 259-286 (2019)
Article DOI: 10.1016/j.ejmech.2019.05.078
BindingDB Entry DOI: 10.7270/Q2ZW1QC8 |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653596
(US11911372, Example 17)Show SMILES COc1ccccc1-c1nnc(NS(=O)(=O)c2c(OC)cccc2OC)s1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 2.07E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653673
(US11911372, Example 96)Show SMILES COCc1ccc(OC)cc1-c1nnc(NS(=O)(=O)c2c(OC)cccc2OC)s1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 2.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653588
(US11911372, Example 9)Show SMILES COc1cccc(c1)-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 2.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653656
(US11911372, Example 78)Show SMILES Cc1ccc(cc1C)S(=O)(=O)Nc1cc(no1)-c1cccc(CCc2ccccc2)c1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 2.51E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653598
(US11911372, Example 19)Show SMILES COc1ccc(CC2CCCCC2)cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 2.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653683
(US11911372, Example 106)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)C(F)(F)F | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 2.86E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653591
(US11911372, Example 12)Show SMILES CCc1ccc(OC)c(c1)S(=O)(=O)Nc1cc(on1)-c1ccc(OC)cc1OC | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653655
(US11911372, Example 77)Show SMILES Cc1ccc(cc1C)S(=O)(=O)Nc1cc(no1)-c1cccc(Cc2ccccc2)c1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 3.27E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653687
(US11911372, Example 110)Show SMILES COc1ccc(Cl)c(c1)-c1nnc(NS(=O)(=O)c2c(OC)cccc2OC)s1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 4.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653589
(US11911372, Example 10)Show SMILES COc1ccccc1-c1cc(NS(=O)(=O)c2c(OC)ccc(-c3ccccc3)c2OC)no1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 5.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653694
(US11911372, Example 117) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 5.26E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653599
(US11911372, Example 20)Show SMILES COc1ccc(CC2CCCCC2)cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)on1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 6.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653679
(US11911372, Example 102) | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 7.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653698
(US11911372, Example 121)Show SMILES COc1ccc(cc1-c1cc(NS(=O)(=O)c2c(OC)cccc2OC)no1)-c1cnn(C)c1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 7.87E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5 Isoform 2 [2-461]
(Homo sapiens (Human)) | BDBM653645
(US11911372, Example 67)Show SMILES Fc1ccc(cc1-c1nnc(NS(=O)(=O)c2ccccc2)s1)-c1ccccc1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| UniChem
| US Patent
| n/a | n/a | 8.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Sumitomo Dainippon Pharma Co., Ltd.
US Patent
| |
US Patent US10815241 (2020)
BindingDB Entry DOI: 10.7270/Q2C82DCF |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM50292429
(2-Hydroxy-6-pentadecyl-benzoic acid | 2-Pentadecyl...)Show InChI InChI=1S/C22H30O3/c1-2-3-4-5-6-7-8-9-10-11-12-13-14-16-19-17-15-18-20(23)21(19)22(24)25/h2,4-5,7-8,15,17-18,23H,1,3,6,9-14,16H2,(H,24,25)/b5-4-,8-7- | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Georgia State University
Curated by ChEMBL
| Assay Description
Inhibition of TIP60 in human HeLa cell extracts by ELISA |
Bioorg Med Chem 17: 1381-6 (2009)
Article DOI: 10.1016/j.bmc.2008.12.014
BindingDB Entry DOI: 10.7270/Q2K35VKS |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM606483
(US11685732, Compound I-130)Show SMILES Cc1cc(cc(C(=O)NNS(=O)(=O)CC2CCOCC2)c1F)-c1cn(C)cn1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
BindingDB Entry DOI: 10.7270/Q28G8QTD |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM606485
(US11685732, Compound I-132)Show SMILES Cc1cc(cc(C(=O)NNS(=O)(=O)CC2CCCN(C2)C(=O)OC(C)(C)C)c1F)-c1cn(C)cn1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
BindingDB Entry DOI: 10.7270/Q28G8QTD |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM606488
(US11685732, Compound I-135)Show SMILES COCCn1cnc(c1)-c1cc(C)c(F)c(c1)C(=O)NNS(=O)(=O)CC1CCCN(C1)C(=O)OC(C)(C)C | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
BindingDB Entry DOI: 10.7270/Q28G8QTD |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM606494
(US11685732, Compound I-141)Show SMILES COCC(=O)N1CCCC(CS(=O)(=O)NNC(=O)c2cc(cc(C)c2F)-c2cn(C)cn2)C1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
BindingDB Entry DOI: 10.7270/Q28G8QTD |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM606495
(US11685732, Compound I-142)Show SMILES CC(=O)N1CCCC(CS(=O)(=O)NNC(=O)c2cc(cc(C)c2F)-c2cn(C)cn2)C1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
BindingDB Entry DOI: 10.7270/Q28G8QTD |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM606510
(US11685732, Compound I-157)Show SMILES Fc1c(Cl)cc(cc1C(=O)NNS(=O)(=O)CC1CCCCC1)-c1ccnn1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
BindingDB Entry DOI: 10.7270/Q28G8QTD |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM606511
(US11685732, Compound I-158)Show SMILES Cn1cc(cn1)-c1cc(Cl)c(F)c(c1)C(=O)NNS(=O)(=O)CC1CCCCC1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
BindingDB Entry DOI: 10.7270/Q28G8QTD |
More data for this
Ligand-Target Pair | |
Histone acetyltransferase KAT5
(Homo sapiens (Human)) | BDBM606512
(US11685732, Compound I-159)Show SMILES Fc1c(Cl)cc(cc1C(=O)NNS(=O)(=O)CC1CCCCC1)-c1cnnc1 | PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
AffyNet
| PC cid
PC sid
UniChem
| | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
| |
Citation and Details
BindingDB Entry DOI: 10.7270/Q28G8QTD |
More data for this
Ligand-Target Pair | |
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