Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260952 (CHEMBL4104489) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50248628 (CHEMBL4072496) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260950 (CHEMBL4100387) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260954 (CHEMBL4070689) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260951 (CHEMBL4077370) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260953 (CHEMBL4072044) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260930 (CHEMBL4087403) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260947 (CHEMBL4095089) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260946 (CHEMBL4077546) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 87 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260959 (CHEMBL4066001) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260961 (CHEMBL4064964) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260955 (CHEMBL4090079) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260929 (CHEMBL4072962) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260927 (CHEMBL4062035) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260948 (CHEMBL4102849) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260928 (CHEMBL4104570) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 410 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260960 (CHEMBL4084901) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 480 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260926 (CHEMBL4082225) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-C/Cyclin-dependent kinase 8 (Homo sapiens (Human)) | BDBM50260949 (CHEMBL4066087) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Medicinal Chemistry, Roche Innovation Center Shanghai, Bldg 5, 720 Cailun Road, Shanghai 201203, China. Electronic address: cyrus.han@roche.com. Curated by ChEMBL | Assay Description Inhibition of recombinant full length His-tagged human CDK8/Cyclin C expressed in baculovirus expression system using Ulight-GS peptide as substrate ... | Bioorg Med Chem Lett 27: 4488-4492 (2017) Article DOI: 10.1016/j.bmcl.2017.07.080 BindingDB Entry DOI: 10.7270/Q2NP26W9 | |||||||||||
More data for this Ligand-Target Pair |