Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583031 (CHEMBL5081078) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 53 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583019 (CHEMBL5081008) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 93 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583020 (CHEMBL5087374) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 130 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583021 (CHEMBL5091289) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 180 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583022 (CHEMBL5085583) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583023 (CHEMBL5081203) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 260 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50220152 ((1S,2R)-2-((S)-Amino-carboxy-methyl)-cyclopropanec...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 262 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2A receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50432711 (CHEMBL2348224) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 277 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2A receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM20180 ((1S,2R,5S,10S,11S,14R,15R)-14-[(2R,5S)-5-hydroxy-6...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 650 | n/a | n/a | n/a | n/a |
SAGE Therapeutics Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as increase in glycine/L-glutama... | J Med Chem 62: 7526-7542 (2019) Article DOI: 10.1021/acs.jmedchem.9b00591 BindingDB Entry DOI: 10.7270/Q2NG4V3J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM18133 (2-aminoacetic acid | CHEMBL773 | Glycine | [14C]Gl...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 990 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM23167 ((2R)-2-amino-3-hydroxypropanoic acid | CHEMBL28512...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50432710 (CHEMBL2348221) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.18E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2A receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM17657 ((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Torino Curated by ChEMBL | Assay Description Agonist activity at rat NR1/NR2A receptor expressed in BHK21 cells assessed as change in intracellular calcium levels by FLIPR assay | J Med Chem 53: 4110-8 (2010) Article DOI: 10.1021/jm1001452 BindingDB Entry DOI: 10.7270/Q2RR206G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583024 (CHEMBL5087170) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583025 (CHEMBL5093773) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.30E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583026 (CHEMBL5072895) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.80E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583027 (CHEMBL5076681) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583028 (CHEMBL5087550) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 6.60E+3 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50531767 (CHEMBL4530995) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.50E+3 | n/a | n/a | n/a | n/a |
University of Bristol Curated by ChEMBL | Assay Description Positive allosteric modulation of rat GluN1/GluN2A expressed in Xenopus laevis oocytes assessed as potentiation of L-glutamate/glycine-induced curren... | Eur J Med Chem 164: 471-498 (2019) Article DOI: 10.1016/j.ejmech.2018.12.054 BindingDB Entry DOI: 10.7270/Q22J6GB9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50461796 (CHEMBL4224777) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a |
Institute of Physiology of the Czech Academy of Sciences Curated by ChEMBL | Assay Description Positive allosteric modulation of recombinant rat GluN1alpha/GluN2A receptor expressed in HEK293 cells assessed as potentiation of glutamate-induced ... | J Med Chem 61: 4505-4516 (2018) Article DOI: 10.1021/acs.jmedchem.8b00255 BindingDB Entry DOI: 10.7270/Q2Z03BTB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583029 (CHEMBL5081696) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+4 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50583030 (CHEMBL5083882) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode volt... | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01810 BindingDB Entry DOI: 10.7270/Q21R6VFZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50531769 (CHEMBL4467653) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.67E+4 | n/a | n/a | n/a | n/a |
University of Bristol Curated by ChEMBL | Assay Description Positive allosteric modulation of rat GluN1/GluN2A expressed in Xenopus laevis oocytes assessed as potentiation of L-glutamate/glycine-induced curren... | Eur J Med Chem 164: 471-498 (2019) Article DOI: 10.1016/j.ejmech.2018.12.054 BindingDB Entry DOI: 10.7270/Q22J6GB9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50503152 (CHEMBL4452216) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.80E+4 | n/a | n/a | n/a | n/a |
University of Bristol Curated by ChEMBL | Assay Description Positive allosteric modulation of rat GluN1/GluN2A expressed in Xenopus laevis oocytes assessed as potentiation of L-glutamate/glycine-induced curren... | Eur J Med Chem 164: 471-498 (2019) Article DOI: 10.1016/j.ejmech.2018.12.054 BindingDB Entry DOI: 10.7270/Q22J6GB9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50432708 (CHEMBL2348223) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | n/a | 2.88E+4 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2A receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50531768 (CHEMBL4531020) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.94E+4 | n/a | n/a | n/a | n/a |
University of Bristol Curated by ChEMBL | Assay Description Positive allosteric modulation of rat GluN1/GluN2A expressed in Xenopus laevis oocytes assessed as potentiation of L-glutamate/glycine-induced curren... | Eur J Med Chem 164: 471-498 (2019) Article DOI: 10.1016/j.ejmech.2018.12.054 BindingDB Entry DOI: 10.7270/Q22J6GB9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50432709 (CHEMBL2348222) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.63E+4 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2A receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50318264 ((+)-2-Amino-3-(4-hydroxy-1,2,5-oxadiazol-3-yl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.70E+4 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Torino Curated by ChEMBL | Assay Description Agonist activity at rat NR1/NR2A receptor expressed in BHK21 cells assessed as change in intracellular calcium levels by FLIPR assay | J Med Chem 53: 4110-8 (2010) Article DOI: 10.1021/jm1001452 BindingDB Entry DOI: 10.7270/Q2RR206G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50318264 ((+)-2-Amino-3-(4-hydroxy-1,2,5-oxadiazol-3-yl)prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4.70E+4 | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Torino Curated by ChEMBL | Assay Description Agonist activity at rat NR1/NR2A receptor expressed in BHK21 cells assessed as change in intracellular calcium levels by FLIPR assay | J Med Chem 53: 4110-8 (2010) Article DOI: 10.1021/jm1001452 BindingDB Entry DOI: 10.7270/Q2RR206G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50252359 ((R,S)-2-amino-2-(1-hydroxy-1H-pyrazol-5-yl)acetic ...) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.20E+4 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat recombinant wild type GluN1/GluN2A receptor expressed in Xenopus laevis oocytes by two electrode voltage clamp technique | J Med Chem 56: 4071-81 (2013) Article DOI: 10.1021/jm400346a BindingDB Entry DOI: 10.7270/Q20G3MHR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1/2A (Rattus norvegicus (Rat)-RAT) | BDBM50531770 (CHEMBL4572997) | PDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.14E+5 | n/a | n/a | n/a | n/a |
University of Bristol Curated by ChEMBL | Assay Description Positive allosteric modulation of rat GluN1/GluN2A expressed in Xenopus laevis oocytes assessed as potentiation of L-glutamate/glycine-induced curren... | Eur J Med Chem 164: 471-498 (2019) Article DOI: 10.1016/j.ejmech.2018.12.054 BindingDB Entry DOI: 10.7270/Q22J6GB9 | |||||||||||
More data for this Ligand-Target Pair |