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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50195259   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Dipeptidyl peptidase 1


(Homo sapiens (Human))		BDBM50195259
PNG
(CHEMBL3898680)
Show SMILES NC1CCCCC1C(=O)N[C@@H](Cc1ccc(cc1)-c1cccc(c1)C#N)C#N |r|
Show InChI InChI=1S/C23H24N4O/c24-14-17-4-3-5-19(12-17)18-10-8-16(9-11-18)13-20(15-25)27-23(28)21-6-1-2-7-22(21)26/h3-5,8-12,20-22H,1-2,6-7,13,26H2,(H,27,28)/t20-,21?,22?/m0/s1
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/a 1.00E+3n/an/an/an/an/an/a



CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED

Curated by ChEMBL


Assay Description
Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assay

J Med Chem 59: 9457-9472 (2016)


Article DOI: 10.1021/acs.jmedchem.6b01127
BindingDB Entry DOI: 10.7270/Q2Z321K4
More data for this
Ligand-Target Pair