Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Epithelial discoidin domain-containing receptor 1 (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.70 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length DDR1 (565 to 876 residues) expressed in bacterial expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epithelial discoidin domain-containing receptor 1 (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 4.70 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length DDR1 (565 to 876 residues) expressed in bacterial expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
NT-3 growth factor receptor (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a |
Jinan University Curated by ChEMBL | Assay Description Binding affinity to TrkC (unknown origin) | J Med Chem 62: 7431-7444 (2019) Article DOI: 10.1021/acs.jmedchem.9b00365 BindingDB Entry DOI: 10.7270/Q2DZ0CSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
NT-3 growth factor receptor (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length TRKC (531 to 825 residues) expressed in mammalian expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
NT-3 growth factor receptor (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length TRKC (531 to 825 residues) expressed in mammalian expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
BDNF/NT-3 growth factors receptor (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a |
Jinan University Curated by ChEMBL | Assay Description Binding affinity to TrkB (unknown origin) | J Med Chem 62: 7431-7444 (2019) Article DOI: 10.1021/acs.jmedchem.9b00365 BindingDB Entry DOI: 10.7270/Q2DZ0CSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
BDNF/NT-3 growth factors receptor (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length TRKB (547 to 838 residues) expressed in mammalian expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
BDNF/NT-3 growth factors receptor (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 22 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length TRKB (547 to 838 residues) expressed in mammalian expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
High affinity nerve growth factor receptor (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length TRKA (475 to 790 residues) expressed in mammalian expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
High affinity nerve growth factor receptor (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length TRKA (475 to 790 residues) expressed in mammalian expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 11B (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length CDK11 (1 to 360 residues) expressed in bacterial expression system preincubated for 1 hr measured ... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 11B (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 370 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length CDK11 (1 to 360 residues) expressed in bacterial expression system preincubated for 1 hr measured ... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscle, skeletal receptor tyrosine-protein kinase (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length MUSK (553 to 869 residues) expressed in bacterial expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Muscle, skeletal receptor tyrosine-protein kinase (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 530 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length MUSK (553 to 869 residues) expressed in bacterial expression system preincubated for 1 hr measured... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ephrin type-A receptor 8 (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length EPHA8 (608 to 920 residues) expressed in bacterial expression system preincubated for 1 hr measure... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Ephrin type-A receptor 8 (Homo sapiens (Human)) | BDBM50528539 (CHEMBL4553037) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 550 | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Sciences Curated by ChEMBL | Assay Description Binding affinity to wild type human partial length EPHA8 (608 to 920 residues) expressed in bacterial expression system preincubated for 1 hr measure... | J Med Chem 59: 5911-6 (2016) Article DOI: 10.1021/acs.jmedchem.6b00140 BindingDB Entry DOI: 10.7270/Q20G3PMX | |||||||||||
More data for this Ligand-Target Pair |