Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine receptor A3 [I248L] (Homo sapiens (Human)) | BDBM191045 (US9181253, 108) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 12.1 | -45.2 | n/a | n/a | n/a | n/a | n/a | 7.5 | 25 |
The United States of America, as represented by the Secretary, Department of Health and Human Services US Patent | Assay Description Radioligand binding assays at A1, A2A, and A3ARs were performed according to the procedures described previously. Each tube in the binding assay cont... | US Patent US9181253 (2015) BindingDB Entry DOI: 10.7270/Q2CV4GJ4 | |||||||||||
More data for this Ligand-Target Pair |