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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Aminopeptidase N' and Ligand = 'BDBM50267841'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Aminopeptidase N


(Sus scrofa (Pig))		BDBM50267841
PNG
((R)-5-Oxo-5-4-[(1,3-thiazole-2-amino)sulfonyl]phen...)
Show SMILES COc1cc(cc(OC)c1OC)C(=O)N[C@H](CCC(O)=O)C(=O)Nc1ccc(cc1)S(=O)(=O)Nc1nccs1 |r|
Show InChI InChI=1S/C24H26N4O9S2/c1-35-18-12-14(13-19(36-2)21(18)37-3)22(31)27-17(8-9-20(29)30)23(32)26-15-4-6-16(7-5-15)39(33,34)28-24-25-10-11-38-24/h4-7,10-13,17H,8-9H2,1-3H3,(H,25,28)(H,26,32)(H,27,31)(H,29,30)/t17-/m1/s1
PDB

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 4.01E+4n/an/an/an/an/an/a



Shandong University

Curated by ChEMBL


Assay Description
Inhibition of pig kidney microsome aminopeptidase N by UV-visible spectrophotometer

Bioorg Med Chem 17: 3053-60 (2009)


Article DOI: 10.1016/j.bmc.2009.02.063
BindingDB Entry DOI: 10.7270/Q2NP25BQ
More data for this
Ligand-Target Pair