Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aryl hydrocarbon receptor (Homo sapiens (Human)) | BDBM50563365 (CHEMBL4750416) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | n/a | n/a | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aryl hydrocarbon receptor (Homo sapiens (Human)) | BDBM50563365 (CHEMBL4750416) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at AHR in human HepG2 cells incubated for 4.5 hrs by Luciferase reporter assay | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113231 BindingDB Entry DOI: 10.7270/Q2NC64XB | |||||||||||
More data for this Ligand-Target Pair |