Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-2 adrenergic receptor (Homo sapiens (Human)) | BDBM50569861 (BI 1744 | CHEBI:82700 | Olodaterol | Striverdi res...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.0871 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at human beta2 adrenoreceptor overexpressed in HEK293 cells assessed as cAMP accumulation | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113697 BindingDB Entry DOI: 10.7270/Q2W95F1H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-2 adrenergic receptor (Homo sapiens (Human)) | BDBM50569861 (BI 1744 | CHEBI:82700 | Olodaterol | Striverdi res...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.0200 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at beta2 adrenoceptor (unknown origin) | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01195 BindingDB Entry DOI: 10.7270/Q24F1VJ7 | |||||||||||
More data for this Ligand-Target Pair |