Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
C-C chemokine receptor type 2 (Homo sapiens (Human)) | BDBM50371414 (CHEMBL271828) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonist activity at human CCR2 in PBMCs assessed as inhibition of chemotaxis | J Med Chem 51: 721-4 (2008) Article DOI: 10.1021/jm701488f BindingDB Entry DOI: 10.7270/Q2TX3G60 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 2 (Homo sapiens (Human)) | BDBM50371414 (CHEMBL271828) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Antagonist activity at human CCR2 in PBMCs assessed as inhibition of MCP1-induced calcium flux | J Med Chem 51: 721-4 (2008) Article DOI: 10.1021/jm701488f BindingDB Entry DOI: 10.7270/Q2TX3G60 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 2 (Homo sapiens (Human)) | BDBM50371414 (CHEMBL271828) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of radiolabeled MCP1 from human CCR2 in PBMCs | J Med Chem 51: 721-4 (2008) Article DOI: 10.1021/jm701488f BindingDB Entry DOI: 10.7270/Q2TX3G60 | |||||||||||
More data for this Ligand-Target Pair |