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Found 1 hit Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM234288'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Cannabinoid receptor 1


(Cricetulus griseus (Chinese hamster))		BDBM234288
PNG
([2-[(5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-m...)
Show SMILES COC(=O)COc1nn(c(c1C)-c1ccc(Cl)cc1)-c1ccc(Cl)cc1Cl
Show InChI InChI=1S/C19H15Cl3N2O3/c1-11-18(12-3-5-13(20)6-4-12)24(16-8-7-14(21)9-15(16)22)23-19(11)27-10-17(25)26-2/h3-9H,10H2,1-2H3
PDB

UniProtKB/TrEMBL

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 182n/an/an/an/an/an/a



NanChang University School of Pharmaceutical Science



Assay Description
The target compounds were evaluated using a binding assay towards the CB1 receptor expressed on the membranes of Chinese hamster ovarian (CHO) cells....

J Enzyme Inhib Med Chem 26: 222-30 (2011)


Article DOI: 10.3109/14756366.2010.491794
BindingDB Entry DOI: 10.7270/Q26D5RW8
More data for this
Ligand-Target Pair