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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Cyclin-C' and Ligand = 'BDBM50567858'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Cyclin-C


(Homo sapiens (Human))		BDBM50567858
PNG
(CHEMBL4878338)
Show SMILES Clc1cncc(-c2ccc(CN3CCOCC3)s2)c1N1CCC2(CCNC2=O)CC1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
 32n/an/an/an/an/an/an/an/a


TBA

Assay Description
Inhibition of CDK8/Cyclin C (unknown origin) using RBER-CHKtide as substrate in presence of [32P]gammaATP incubated for 60 mins by microplate scintil...

Citation and Details

Article DOI: 10.1016/j.ejmech.2021.113391
BindingDB Entry DOI: 10.7270/Q29P35DW
More data for this
Ligand-Target Pair