BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Cytosol aminopeptidase [33-68,L62W]' and Ligand = 'BDBM234298'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Cytosol aminopeptidase [33-68,L62W]


(Sus scrofa (Pig))		BDBM234298
PNG
(Nle-ψ[P(O)(OH)O]-L-Ala (6))
Show SMILES CCCCC(N)P(O)(=O)O[C@@H](C)C(O)=O |r|
Show InChI InChI=1S/C8H18NO5P/c1-3-4-5-7(9)15(12,13)14-6(2)8(10)11/h6-7H,3-5,9H2,1-2H3,(H,10,11)(H,12,13)/t6-,7?/m0/s1
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
 2.69E+5 -20.4n/an/an/an/an/a8.425



Academy of Sciences of the Czech Republic



Assay Description
LAP was assayed in 75 mM triethanolamine hydrochloride buffer (pH = 8.4, containing 5 mM MgCl2) at 25°C. The substrate (L-leucine-p-nitroanilide) was...

J Enzyme Inhib Med Chem 26: 155-61 (2011)


Article DOI: 10.3109/14756366.2010.482047
BindingDB Entry DOI: 10.7270/Q22N515B
More data for this
Ligand-Target Pair