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Found 1 hit Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 9' and Ligand = 'BDBM50359367'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Dipeptidyl peptidase 9


(Homo sapiens (Human))		BDBM50359367
PNG
(CHEMBL1929388)
Show SMILES Cc1cc2ncc(C(=O)NCC(C)(C)NCC(=O)N3CCC[C@H]3C#N)c(C)n2n1 |r|
Show InChI InChI=1S/C20H27N7O2/c1-13-8-17-22-10-16(14(2)27(17)25-13)19(29)23-12-20(3,4)24-11-18(28)26-7-5-6-15(26)9-21/h8,10,15,24H,5-7,11-12H2,1-4H3,(H,23,29)/t15-/m0/s1
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Article
PubMed
n/an/a 64n/an/an/an/an/an/a



Sanwa Kagaku Kenkyusho Co. Ltd

Curated by ChEMBL


Assay Description
Inhibition of human recombinant DPP-9 expressed in Sf9 cells using H-Gly-Pro-AMC as substrate preincubated for 30 mins before substrate addition meas...

Bioorg Med Chem 19: 7221-7 (2011)


Article DOI: 10.1016/j.bmc.2011.09.043
BindingDB Entry DOI: 10.7270/Q2862GVX
More data for this
Ligand-Target Pair