Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Egl nine homolog 1 (Homo sapiens (Human)) | BDBM93411 (PHD Inhibitor, 8{1}) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 482 | n/a | n/a | n/a | n/a | n/a | n/a |
Amgen, Inc. | Assay Description PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI... | J Comb Chem 12: 676-86 (2010) Article DOI: 10.1021/cc100073a BindingDB Entry DOI: 10.7270/Q2B27SXP | |||||||||||
More data for this Ligand-Target Pair |