Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gamma-aminobutyric acid receptor subunit alpha-2 (Rattus norvegicus (Rat)) | BDBM50044427 (1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]hexade...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Tested for invitro inhibition of the displacement of [3H]-mazindol from GABA receptor | J Med Chem 36: 2499-507 (1993) BindingDB Entry DOI: 10.7270/Q2V69HNK | |||||||||||
More data for this Ligand-Target Pair |