Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50002695 (7,8-Dichloro-5H-1,2,3,5,9b-pentaaza-cyclopenta[a]n...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Lilly Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]glycine from glycine site on the NMDA receptor. | J Med Chem 35: 3319-24 (1992) BindingDB Entry DOI: 10.7270/Q2WM1F13 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50002695 (7,8-Dichloro-5H-1,2,3,5,9b-pentaaza-cyclopenta[a]n...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 7.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Compound was evaluated for its binding affinity towards strychnine - insensitive glycine site of NMDA receptor in presence of [3H]- Gly | Bioorg Med Chem Lett 1: 751-756 (1991) Article DOI: 10.1016/S0960-894X(01)81062-3 BindingDB Entry DOI: 10.7270/Q2J67GTV | |||||||||||
More data for this Ligand-Target Pair |