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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1' and Ligand = 'BDBM50082020'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glutamate receptor ionotropic, NMDA 1


(RAT)		BDBM50082020
PNG
(2-Chloro-N-{2-[3-(7-chloro-4-hydroxy-2-oxo-1,2-dih...)
Show SMILES Oc1c(-c2cccc(Oc3ccccc3NC(=O)CCl)c2)c(=O)[nH]c2cc(Cl)ccc12
Show InChI InChI=1S/C23H16Cl2N2O4/c24-12-20(28)26-17-6-1-2-7-19(17)31-15-5-3-4-13(10-15)21-22(29)16-9-8-14(25)11-18(16)27-23(21)30/h1-11H,12H2,(H,26,28)(H2,27,29,30)
PDB

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem

Similars
PubMed
 7.10n/an/an/an/an/an/an/an/a



Université Louis Pasteur

Curated by ChEMBL


Assay Description
Displacement of [3H]-5-7 dichlorokynurenic acid ([3H]- DCKA) from N-methyl-D-aspartate glutamate receptor glycine site of rat brain membrane homogen...

J Med Chem 42: 4394-404 (1999)


BindingDB Entry DOI: 10.7270/Q2HT2NJB
More data for this
Ligand-Target Pair