BindingDB PrimarySearch

Found 9 hits Enz. Inhib. hit(s) with Target = 'Glycogen phosphorylase, muscle form' and Ligand = 'BDBM50295860'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	7.60E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Debrecen Curated by ChEMBL					Assay Description Inhibition of rabbit muscle glycogen phosphorylase b				ACS Med Chem Lett 4: 612-5 (2013) Article DOI: 10.1021/ml4001529 BindingDB Entry DOI: 10.7270/Q2X068FD
University of Debrecen Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	7.60E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Debrecen Curated by ChEMBL					Assay Description Inhibition of rabbit muscle glycogen phosphorylase b				Eur J Med Chem 76: 567-79 (2014) Article DOI: 10.1016/j.ejmech.2014.02.041 BindingDB Entry DOI: 10.7270/Q2ZP47N4
University of Debrecen Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	7.60E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Debrecen Curated by ChEMBL					Assay Description Competitive inhibition of rabbit muscle glycogen phosphorylase-b using glucose-1-phosphate as substrate preincubated with glycogen for 15 mins follow...				ACS Med Chem Lett 6: 1215-9 (2015) Article DOI: 10.1021/acsmedchemlett.5b00361 BindingDB Entry DOI: 10.7270/Q2W37Z56
University of Debrecen Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	7.60E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Debrecen Curated by ChEMBL					Assay Description Inhibition of rabbit muscle glycogen phosphorylase b				Bioorg Med Chem 17: 4773-85 (2009) Article DOI: 10.1016/j.bmc.2009.04.036 BindingDB Entry DOI: 10.7270/Q2Q52PPV
University of Debrecen Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	7.60E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Egypt National Research Centre Curated by ChEMBL					Assay Description Inhibition of rabbit skeletal muscle glycogen phosphorylase b assessed as inorganic phosphate release using glucose-1-phosphate as substrate by doubl...				Bioorg Med Chem 24: 5423-5430 (2016) Article DOI: 10.1016/j.bmc.2016.08.069 BindingDB Entry DOI: 10.7270/Q26D5VZD
Egypt National Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	7.60E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Thessaly Curated by ChEMBL					Assay Description Competitive inhibition of rabbit muscle glycogen phosphorylase-b in presence of varying levels of glucose-1-phosphate and constant concentration of g...				Eur J Med Chem 123: 737-745 (2016) Article DOI: 10.1016/j.ejmech.2016.06.049 BindingDB Entry DOI: 10.7270/Q2TT4SXG
University of Thessaly Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	2.29E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Thessaly Curated by ChEMBL					Assay Description Inhibition of rabbit muscle glycogen phosphorylase-b				Eur J Med Chem 123: 737-745 (2016) Article DOI: 10.1016/j.ejmech.2016.06.049 BindingDB Entry DOI: 10.7270/Q2TT4SXG
University of Thessaly Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	2.29E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Egypt National Research Centre Curated by ChEMBL					Assay Description Inhibition of rabbit muscle glycogen phosphorylase b using alpha-D-glucose-1-phosphate as substrate				Bioorg Med Chem 24: 5423-5430 (2016) Article DOI: 10.1016/j.bmc.2016.08.069 BindingDB Entry DOI: 10.7270/Q26D5VZD
Egypt National Research Centre Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Glycogen phosphorylase, muscle form (Oryctolagus cuniculus (rabbit))	BDBM50295860 ((2R,3R,4S,5S,6R)-2-(benzo[d]thiazol-2-yl)-6-(hydro...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet	CHEMBL MMDB PC cid PC sid PDB UniChem	MMDB PDB Article PubMed	2.29E+5	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
University of Debrecen Curated by ChEMBL					Assay Description Inhibition of rabbit muscle glycogen phosphorylase-b				ACS Med Chem Lett 6: 1215-9 (2015) Article DOI: 10.1021/acsmedchemlett.5b00361 BindingDB Entry DOI: 10.7270/Q2W37Z56
University of Debrecen Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)