Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Heat sensitive channel TRPV3 (Rattus norvegicus) | BDBM50535865 (CHEMBL4543647) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
National Research Council Curated by ChEMBL | Assay Description Antagonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as inhibition of thymol-induced intracellular calcium accumulation pr... | J Med Chem 59: 5661-83 (2016) Article DOI: 10.1021/acs.jmedchem.5b01448 BindingDB Entry DOI: 10.7270/Q2222Z8V | |||||||||||
More data for this Ligand-Target Pair |