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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM22904 ((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...) | UniProtKB/SwissProt GoogleScholar AffyNet  | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Queen's Medical Centre Curated by PDSP Ki Database | Biochem Soc Trans 20: 122-5 (1992) Article DOI: 10.1042/bst0200122 BindingDB Entry DOI: 10.7270/Q2RX99KH | ||||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM22904 ((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Binding afinity against H1 receptor | J Med Chem 38: 1593-9 (1995) BindingDB Entry DOI: 10.7270/Q2BK1BC1 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histamine H1 receptor (Cavia porcellus (domestic guinea pig)) | BDBM22904 ((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Schering-Plough Research Institute Curated by ChEMBL | Assay Description Binding affinity of the compound to H-1 receptor was determined in guinea pig brain tissue using [3H]- N alpha-methylhistamine ligand | Bioorg Med Chem Lett 8: 243-8 (1999) BindingDB Entry DOI: 10.7270/Q2ST7P0Z | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
