Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50146232 (CHEMBL440696 | Phosphoric acid mono-{(R)-2-((Z)-oc...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Virginia Curated by ChEMBL | Assay Description In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell lines | Bioorg Med Chem Lett 14: 2735-40 (2004) Article DOI: 10.1016/j.bmcl.2004.03.076 BindingDB Entry DOI: 10.7270/Q2DF6QN9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50146232 (CHEMBL440696 | Phosphoric acid mono-{(R)-2-((Z)-oc...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Virginia Curated by ChEMBL | Assay Description Binding affinity towards Lysophosphatidic acid 1 (LPA1) receptor | Bioorg Med Chem Lett 14: 4069-74 (2004) Article DOI: 10.1016/j.bmcl.2004.05.023 BindingDB Entry DOI: 10.7270/Q2930SM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50146232 (CHEMBL440696 | Phosphoric acid mono-{(R)-2-((Z)-oc...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 109 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Virginia Curated by ChEMBL | Assay Description Inhibitory concentration against Lysophosphatidic acid 1 (LPA1) receptor | Bioorg Med Chem Lett 14: 4069-74 (2004) Article DOI: 10.1016/j.bmcl.2004.05.023 BindingDB Entry DOI: 10.7270/Q2930SM1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50146232 (CHEMBL440696 | Phosphoric acid mono-{(R)-2-((Z)-oc...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 109 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Virginia Curated by ChEMBL | Assay Description In vitro ability to antagonize LPA-evoked [35S]-GTP-gammaS binding to lysophosphatidic acid receptor 1 in HEK293T cell lines | Bioorg Med Chem Lett 14: 2735-40 (2004) Article DOI: 10.1016/j.bmcl.2004.03.076 BindingDB Entry DOI: 10.7270/Q2DF6QN9 | |||||||||||
More data for this Ligand-Target Pair |