Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Lysophosphatidic acid receptor 1 (Homo sapiens (Human)) | BDBM50517246 (CHEMBL4557434) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Therachem Research Medilab, LLC Curated by ChEMBL | Assay Description Antagonist activity at human LPA1 expressed in CHO cells assessed as reduction in LPA-induced calcium influx incubated for 20 mins | ACS Med Chem Lett 10: 1378-1379 (2019) Article DOI: 10.1021/acsmedchemlett.9b00429 BindingDB Entry DOI: 10.7270/Q2GF0XVT | |||||||||||
More data for this Ligand-Target Pair |