Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melatonin receptor type 1C (Gallus gallus) | BDBM85065 (CAS_117946-91-5 | Luzindole | NSC_122162) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 1.61E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University College London Curated by ChEMBL | Assay Description Binding affinity towards melatonin receptor, determined in chicken brain membranes using [2-125I]melatonin | J Med Chem 41: 451-67 (1998) Article DOI: 10.1021/jm970246n BindingDB Entry DOI: 10.7270/Q2154KSH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM85065 (CAS_117946-91-5 | Luzindole | NSC_122162) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 2.04E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
King's College London Curated by PDSP Ki Database | Naunyn Schmiedebergs Arch Pharmacol 358: 522-8 (1998) Article DOI: 10.1007/pl00005288 BindingDB Entry DOI: 10.7270/Q2WW7G6S | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM85065 (CAS_117946-91-5 | Luzindole | NSC_122162) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair |