Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50446953 (CHEMBL3115774) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
Florida Institute of Technology Curated by ChEMBL | Assay Description Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of calcium mobilization by fluorescence assay | ACS Med Chem Lett 5: 815-9 (2014) Article DOI: 10.1021/ml500161v BindingDB Entry DOI: 10.7270/Q2H70HHM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50446953 (CHEMBL3115774) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7 | n/a | n/a | n/a | n/a | n/a | n/a |
McGill University Curated by ChEMBL | Assay Description Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil... | J Med Chem 57: 364-77 (2014) Article DOI: 10.1021/jm401292m BindingDB Entry DOI: 10.7270/Q2N87C82 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50446953 (CHEMBL3115774) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Florida Institute of Technology Curated by ChEMBL | Assay Description Antagonist activity at OXE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobilization incubated for 2 mins follow... | J Med Chem 61: 5934-5948 (2018) Article DOI: 10.1021/acs.jmedchem.8b00154 BindingDB Entry DOI: 10.7270/Q22F7R48 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50446953 (CHEMBL3115774) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Florida Institute of Technology Curated by ChEMBL | Assay Description Antagonist activity at 5-oxo-ETE receptor in human neutrophils assessed as inhibition of 5-oxo-ETE-induced Ca2+ mobilization incubated for 2 mins pri... | Bioorg Med Chem Lett 24: 3385-8 (2014) Article DOI: 10.1016/j.bmcl.2014.05.090 BindingDB Entry DOI: 10.7270/Q2G162F7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50446953 (CHEMBL3115774) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
McGill University Curated by ChEMBL | Assay Description Antagonist activity at OXE receptor (unknown origin) expressed in anti-CD49d-labeled eosinophils assessed as inhibition of 5-oxo-ETE-induced F-actin ... | J Med Chem 57: 364-77 (2014) Article DOI: 10.1021/jm401292m BindingDB Entry DOI: 10.7270/Q2N87C82 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50446953 (CHEMBL3115774) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 402 | n/a | n/a | n/a | n/a | n/a | n/a |
McGill University Curated by ChEMBL | Assay Description Antagonist activity at OXE receptor (unknown origin) expressed in neutrophils assessed as inhibition of 5-oxo-ETE-induced cell migration after 2 hrs ... | J Med Chem 57: 364-77 (2014) Article DOI: 10.1021/jm401292m BindingDB Entry DOI: 10.7270/Q2N87C82 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50446953 (CHEMBL3115774) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
McGill University Curated by ChEMBL | Assay Description Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil... | J Med Chem 57: 364-77 (2014) Article DOI: 10.1021/jm401292m BindingDB Entry DOI: 10.7270/Q2N87C82 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Oxoeicosanoid receptor 1 (Homo sapiens (Human)) | BDBM50446953 (CHEMBL3115774) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
McGill University Curated by ChEMBL | Assay Description Antagonist activity at OXE receptor (unknown origin) expressed in indo-1 loaded neutrophils assessed as inhibition of 5-oxo-ETE-induced calcium mobil... | J Med Chem 57: 364-77 (2014) Article DOI: 10.1021/jm401292m BindingDB Entry DOI: 10.7270/Q2N87C82 | |||||||||||
More data for this Ligand-Target Pair |