Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 14.6 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to against methicillin-, daptomycin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 25 PBP2a by co... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 233 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Notre Dame Curated by ChEMBL | Assay Description Inhibition of methicillin-resistant Staphylococcus aureus PBP 2a | Antimicrob Agents Chemother 53: 4051-63 (2009) Article DOI: 10.1128/AAC.00084-09 BindingDB Entry DOI: 10.7270/Q2R21479 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 365 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, vancomycin-resistant, beta-lactamase-positive Staphylococcus aureus 510 PBP2a by competitive binding assay | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 730 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, heteroresistant vancomycin-intermediate, beta-lactamase-negative Staphylococcus aureus 873 PBP2a by compet... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-, linezolid-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 2149A PBP2a by competit... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptidase (Staphylococcus aureus) | BDBM50482776 (CHEBI:70718 | Ceftaroline Fosamil | PPI-0903 | TAK...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hershey Medical Center Curated by ChEMBL | Assay Description Binding affinity to methicillin-resistant, vancomycin-intermediate, beta-lactamase-positive Staphylococcus aureus 1287 PBP2a by competitive binding a... | Antimicrob Agents Chemother 54: 1670-7 (2010) Article DOI: 10.1128/AAC.00019-10 BindingDB Entry DOI: 10.7270/Q2B56NK6 | |||||||||||
More data for this Ligand-Target Pair |