Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Phosphoglycerate kinase 1 (Homo sapiens (Human)) | BDBM14487 ((2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 3.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington Curated by ChEMBL | Assay Description evaluated for the inhibition of Trypanosoma brucei Phosphoglycerate kinase (PGK) | J Med Chem 43: 4135-50 (2000) Article DOI: 10.1021/jm000287a BindingDB Entry DOI: 10.7270/Q2TB19N4 | |||||||||||
More data for this Ligand-Target Pair |