BindingDB PrimarySearch

Found 9 hits Enz. Inhib. hit(s) with Target = 'Phospholipase A2' and Ligand = 'BDBM50250399'
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Phospholipase A2 (Apis mellifera)	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
University of California-San Diego Curated by ChEMBL					Assay Description Inhibition of bee venom PLA2				J Nat Prod 55: 1701-17 (1992) Article DOI: 10.1021/np50090a001 BindingDB Entry DOI: 10.7270/Q2H70JMC
University of California-San Diego Curated by ChEMBL					More data for this Ligand-Target Pair
Phospholipase A2 (Apis mellifera)	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
Muséum National d'Histoire Naturelle Curated by ChEMBL					Assay Description Inhibition of bee venom phospholipase A2 after 5 mins by spectrophotometric analysis				Bioorg Med Chem 18: 6006-11 (2010) Article DOI: 10.1016/j.bmc.2010.06.066 BindingDB Entry DOI: 10.7270/Q24F1QXH
Muséum National d'Histoire Naturelle Curated by ChEMBL					More data for this Ligand-Target Pair
Phospholipase A2 (Apis mellifera)	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	500	n/a	n/a	n/a	n/a	n/a	n/a
University of Auckland Curated by ChEMBL					Assay Description Inhibition of bee venom phospholipase A2 after 5 mins by spectrophotometric analysis				Bioorg Med Chem Lett 21: 1261-4 (2011) Article DOI: 10.1016/j.bmcl.2010.12.056 BindingDB Entry DOI: 10.7270/Q2125SZK
University of Auckland Curated by ChEMBL					More data for this Ligand-Target Pair
Phospholipase A2 (Homo sapiens (Human))	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Napoli"Federico II" Curated by ChEMBL					Assay Description Inhibition of human synovial secretory PLA2				J Nat Prod 61: 571-5 (1998) Article DOI: 10.1021/np9704922 BindingDB Entry DOI: 10.7270/Q2M32WN8
					More data for this Ligand-Target Pair
Phospholipase A2 (Apis mellifera)	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ degli Studi di Napoli"Federico II" Curated by ChEMBL					Assay Description Inhibition of bee venom secretory PLA2				J Nat Prod 61: 571-5 (1998) Article DOI: 10.1021/np9704922 BindingDB Entry DOI: 10.7270/Q2M32WN8
					More data for this Ligand-Target Pair
Phospholipase A2 (Apis mellifera)	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	7.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
Università degli Studi di Napoli Federico II Curated by ChEMBL					Assay Description Inhibition of bee venom group 3 secretory phospholipase A2 by liquid scintillation counting				J Nat Prod 64: 612-5 (2001) BindingDB Entry DOI: 10.7270/Q28915MQ
					More data for this Ligand-Target Pair
Phospholipase A2 (Apis mellifera)	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
Istituto per la Chimica di Molecole di Interesse Biologico CNR Curated by ChEMBL					Assay Description Inhibition of bee venom group3 sPLA2 by liquid scintillation counting				J Nat Prod 61: 931-5 (1998) Article DOI: 10.1021/np980122t BindingDB Entry DOI: 10.7270/Q2BK1D8H
					More data for this Ligand-Target Pair
Phospholipase A2 (Apis mellifera)	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universit£ di Salerno Curated by ChEMBL					Assay Description Inhibitory activity against bee secretory Phospholipase A2 enzyme				J Med Chem 41: 3232-8 (1998) Article DOI: 10.1021/jm980027h BindingDB Entry DOI: 10.7270/Q2ZP46SH
Universit£ di Salerno Curated by ChEMBL					More data for this Ligand-Target Pair
Phospholipase A2 (Apis mellifera)	BDBM50250399 (5-Hydroxy-4-{(R)-6-hydroxy-5-[(E)-4-methyl-6-(2,6,...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.25E+4	n/a	n/a	n/a	n/a	n/a	n/a
Istituto per la Chimica di Molecole di Interesse Biologico CNR Curated by ChEMBL					Assay Description Inhibition of bee venom group3 sPLA2 at 10 uM by liquid scintillation counting				J Nat Prod 61: 931-5 (1998) Article DOI: 10.1021/np980122t BindingDB Entry DOI: 10.7270/Q2BK1D8H
					More data for this Ligand-Target Pair