BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50018324'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50018324
PNG
(CHEMBL299760 | [1,1';2',1'']Terphenyl-4'-carboxyli...)
Show SMILES C[C@H](CCCc1cccnc1)NC(=O)c1ccc(-c2ccccc2)c(c1)-c1ccccc1
Show InChI InChI=1S/C29H28N2O/c1-22(10-8-11-23-12-9-19-30-21-23)31-29(32)26-17-18-27(24-13-4-2-5-14-24)28(20-26)25-15-6-3-7-16-25/h2-7,9,12-22H,8,10-11H2,1H3,(H,31,32)/t22-/m1/s1
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars
PubMed
n/an/a 50n/an/an/an/an/an/a



Roche Research Center

Curated by ChEMBL


Assay Description
Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.

J Med Chem 32: 1814-20 (1989)


BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ
More data for this
Ligand-Target Pair