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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50018329'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50018329
PNG
(3',4'-Dimethoxy-biphenyl-4-carbothioic acid (1-met...)
Show SMILES COc1ccc(cc1OC)-c1ccc(cc1)C(=S)N[C@H](C)CCCc1cccnc1
Show InChI InChI=1S/C25H28N2O2S/c1-18(6-4-7-19-8-5-15-26-17-19)27-25(30)21-11-9-20(10-12-21)22-13-14-23(28-2)24(16-22)29-3/h5,8-18H,4,6-7H2,1-3H3,(H,27,30)/t18-/m1/s1
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Roche Research Center

Curated by ChEMBL


Assay Description
Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.

J Med Chem 32: 1814-20 (1989)


BindingDB Entry DOI: 10.7270/Q2SQ8ZCJ
More data for this
Ligand-Target Pair