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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-activating factor receptor' and Ligand = 'BDBM50018394'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-activating factor receptor


(Homo sapiens (Human))		BDBM50018394
PNG
(5,5-Bis-(3,4-dimethoxy-phenyl)-penta-2,4-dienoic a...)
Show SMILES [#6]-[#8]-c1ccc(cc1-[#8]-[#6])-[#6](=[#6]/[#6]=[#6]/[#6](=O)-[#7]-[#6@H](-[#6])-[#6]-[#6]-[#6]-c1cccnc1)\c1ccc(-[#8]-[#6])c(-[#8]-[#6])c1
Show InChI InChI=1S/C31H36N2O5/c1-22(9-6-10-23-11-8-18-32-21-23)33-31(34)13-7-12-26(24-14-16-27(35-2)29(19-24)37-4)25-15-17-28(36-3)30(20-25)38-5/h7-8,11-22H,6,9-10H2,1-5H3,(H,33,34)/b13-7+/t22-/m1/s1
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PubMed
n/an/a 50n/an/an/an/an/an/a



Roche Research Center

Curated by ChEMBL


Assay Description
Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand

J Med Chem 32: 1820-35 (1989)


BindingDB Entry DOI: 10.7270/Q2NZ86MR
More data for this
Ligand-Target Pair