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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Platelet-derived growth factor receptor beta' and Ligand = 'BDBM4850'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Platelet-derived growth factor receptor beta


(Homo sapiens (Human))		BDBM4850
PNG
(1-{2-amino-6-[3,5-bis(dimethylamino)phenyl]pyrido[...)
Show SMILES CN(C)c1cc(cc(c1)-c1cc2cnc(N)nc2nc1NC(=O)NC(C)(C)C)N(C)C
Show InChI InChI=1S/C22H30N8O/c1-22(2,3)28-21(31)27-19-17(10-14-12-24-20(23)26-18(14)25-19)13-8-15(29(4)5)11-16(9-13)30(6)7/h8-12H,1-7H3,(H4,23,24,25,26,27,28,31)
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Similars
Article
n/an/a>5.00E+4n/an/an/an/an/an/a



Parke-Davis Pharmaceutical Research



Assay Description
The kinase activity is the enzyme activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ATP to the poly (E: Y) substrate. N...

Bioorg Med Chem Lett 7: 2415-20 (1997)


Article DOI: 10.1074/jbc.M606873200
BindingDB Entry DOI: 10.7270/Q28C9TF2
More data for this
Ligand-Target Pair