Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Polyamine deacetylase HDAC10 (Homo sapiens (Human)) | BDBM50398716 (CHEMBL2179618 | US10227295, Compound 5g | US940985...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
European Molecular Biology Laboratory Curated by ChEMBL | Assay Description Inhibition of tubastatin-Alexa647-tracer binding to recombinant GST-tagged HDAC10 (unknown origin) measured after 1 hr by TR-FRET assay | J Med Chem 62: 4426-4443 (2019) Article DOI: 10.1021/acs.jmedchem.8b01936 BindingDB Entry DOI: 10.7270/Q26H4MTC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polyamine deacetylase HDAC10 (Homo sapiens (Human)) | BDBM50398716 (CHEMBL2179618 | US10227295, Compound 5g | US940985...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 501 | n/a | n/a | n/a | n/a | n/a | n/a |
European Molecular Biology Laboratory Curated by ChEMBL | Assay Description Inhibition of dye-labeled tracer binding to HDAC10 (unknown origin) transfected in human HeLa cells measured after 2 hrs by nano-luciferase reporter ... | J Med Chem 62: 4426-4443 (2019) Article DOI: 10.1021/acs.jmedchem.8b01936 BindingDB Entry DOI: 10.7270/Q26H4MTC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polyamine deacetylase HDAC10 (Homo sapiens (Human)) | BDBM50398716 (CHEMBL2179618 | US10227295, Compound 5g | US940985...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 7.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Illinois at Chicago Curated by ChEMBL | Assay Description Inhibition of HDAC10 | J Med Chem 55: 9891-9 (2012) Article DOI: 10.1021/jm301098e BindingDB Entry DOI: 10.7270/Q2WQ04XP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Polyamine deacetylase HDAC10 (Homo sapiens (Human)) | BDBM50398716 (CHEMBL2179618 | US10227295, Compound 5g | US940985...) | NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 7.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of HDAC10 (unknown origin) | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113526 BindingDB Entry DOI: 10.7270/Q2D79G8J | |||||||||||
More data for this Ligand-Target Pair |