Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prostaglandin E2 receptor EP3 subtype (Homo sapiens (Human)) | BDBM50248275 (CHEMBL474751 | N-(3,4-difluorophenylsulfonyl)-3-(1...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a |
deCODE Chemistry Curated by ChEMBL | Assay Description Displacement of [3H]PGE2 from human EP3 receptor at 20 uM in presence of normal buffer | Bioorg Med Chem Lett 19: 1528-31 (2009) Article DOI: 10.1016/j.bmcl.2008.12.112 BindingDB Entry DOI: 10.7270/Q2JM29H0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin E2 receptor EP3 subtype (Homo sapiens (Human)) | BDBM50248275 (CHEMBL474751 | N-(3,4-difluorophenylsulfonyl)-3-(1...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
deCODE Chemistry Curated by ChEMBL | Assay Description Displacement of [3H]PGE2 from human EP3 receptor at 20 uM in presence of 10% human serum | Bioorg Med Chem Lett 19: 1528-31 (2009) Article DOI: 10.1016/j.bmcl.2008.12.112 BindingDB Entry DOI: 10.7270/Q2JM29H0 | |||||||||||
More data for this Ligand-Target Pair |