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Found 1 hit Enz. Inhib. hit(s) with Target = 'Proto-oncogene Wnt-1' and Ligand = 'BDBM384771'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Proto-oncogene Wnt-1


(Homo sapiens (human))		BDBM384771
PNG
(US10285983, Compound 271)
Show SMILES CCCCC(=O)Nc1cncc(c1)-c1cnc2[nH]nc(-c3cc4cccnc4[nH]3)c2c1
Show InChI InChI=1S/C23H21N7O/c1-2-3-6-20(31)27-17-8-15(11-24-13-17)16-9-18-21(29-30-23(18)26-12-16)19-10-14-5-4-7-25-22(14)28-19/h4-5,7-13H,2-3,6H2,1H3,(H,25,28)(H,27,31)(H,26,29,30)
UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a>1.00E+4n/an/an/an/a



Istanbul University



Assay Description
SW480 colon carcinoma cells were transduced with a lentiviral vector expressing luciferase with a human Sp5 promoter consisting of a sequence of eigh...

Bioorg Med Chem 16: 9113-20 (2008)


BindingDB Entry DOI: 10.7270/Q2D79DQJ
More data for this
Ligand-Target Pair