Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Queuine tRNA-ribosyltransferase (Zymomonas mobilis) | BDBM84652 (Quinazolinone scaffold, 1) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | 7.3 | n/a |
Philipps-Universität Marburg | Assay Description Inhibition assay using tRNA-guanine transglycosylase (TGT). | Chembiochem 10: 716-27 (2009) Article DOI: 10.1002/cbic.200800782 BindingDB Entry DOI: 10.7270/Q20R9MX5 | |||||||||||
More data for this Ligand-Target Pair |