Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase N1 (Homo sapiens (Human)) | BDBM50545100 (CHEMBL1990482) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sussex Curated by ChEMBL | Assay Description Displacement of tracer from PKN1 (unknown origin) by TR-FRET assay | Bioorg Med Chem Lett 30: (2020) Article DOI: 10.1016/j.bmcl.2020.127040 BindingDB Entry DOI: 10.7270/Q2SJ1Q61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase N1 (Homo sapiens (Human)) | BDBM50545100 (CHEMBL1990482) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | <1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sussex Curated by ChEMBL | Assay Description Inhibition of His/GST-tagged PKN1 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo... | Bioorg Med Chem Lett 30: (2020) Article DOI: 10.1016/j.bmcl.2020.127040 BindingDB Entry DOI: 10.7270/Q2SJ1Q61 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase N1 (Homo sapiens (Human)) | BDBM50545100 (CHEMBL1990482) | PDB MMDB NCI pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sussex Curated by ChEMBL | Assay Description Displacement of tracer from PKN1 (unknown origin) by TR-FRET assay | Bioorg Med Chem Lett 30: (2020) Article DOI: 10.1016/j.bmcl.2020.127040 BindingDB Entry DOI: 10.7270/Q2SJ1Q61 | |||||||||||
More data for this Ligand-Target Pair |