Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sigma non-opioid intracellular receptor 1 (RAT) | BDBM50000663 ((+)-1-methyl-16-azatetracyclo[7.6.1.02,7.010,15]he...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 5.92E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Tested for invitro inhibition of the displacement of (+)-[3H]-pentazocine from sigma opioid receptor | J Med Chem 36: 2499-507 (1993) BindingDB Entry DOI: 10.7270/Q2V69HNK | |||||||||||
More data for this Ligand-Target Pair |