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Found 1 hit Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 2 subunit alpha' and Ligand = 'BDBM50107051'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Sodium channel protein type 2 subunit alpha


(Homo sapiens (Human))		BDBM50107051
PNG
(CHEMBL108627 | N-(4-Methyl-benzoyl)-N'-naphthalen-...)
Show SMILES Cc1ccc(cc1)C(=O)NC(N)=NCc1cccc2ccccc12 |w:12.13|
Show InChI InChI=1S/C20H19N3O/c1-14-9-11-16(12-10-14)19(24)23-20(21)22-13-17-7-4-6-15-5-2-3-8-18(15)17/h2-12H,13H2,1H3,(H3,21,22,23,24)
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PubMed
n/an/a 2.38E+3n/an/an/an/an/an/a



CeNeS Pharmaceuticals Inc.

Curated by ChEMBL


Assay Description
Inhibition of sodium channel blockade in CHO cells expressing neuronal mammalian type IIA (CNaIIA) sodium channel

Bioorg Med Chem Lett 11: 3151-5 (2001)


BindingDB Entry DOI: 10.7270/Q2PC31P4
More data for this
Ligand-Target Pair