Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Solute carrier organic anion transporter family member 1A4 (Rattus norvegicus) | BDBM50375594 (TAUROCHOLATE) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | PubMed | 3.94E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of E217betaG uptake in Oatp2-expressing LLC-PK1 cells | J Pharmacol Exp Ther 298: 316-22 (2001) BindingDB Entry DOI: 10.7270/Q2XW4M2T | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier organic anion transporter family member 1A4 (Rattus norvegicus) | BDBM50375594 (TAUROCHOLATE) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | PubMed | 1.56E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
the University of Tokyo Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Digoxin uptake in Oatp2-expressing LLC-PK1 cells | Drug Metab Dispos 30: 220-3 (2002) BindingDB Entry DOI: 10.7270/Q22N53J3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier organic anion transporter family member 1A4 (Rattus norvegicus) | BDBM50375594 (TAUROCHOLATE) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG MMDB PC cid PC sid PDB UniChem Similars | PubMed | n/a | n/a | 1.48E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kyoto University Hospital Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Digoxin uptake in Xenopus laevis oocytes | J Pharmacol Exp Ther 299: 261-7 (2001) BindingDB Entry DOI: 10.7270/Q2JS9RQF | |||||||||||
More data for this Ligand-Target Pair |