Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50457473 (CHEMBL4209822) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Jadavpur University Curated by ChEMBL | Assay Description Inhibition of porcine kidney leucine aminopeptidase using LGG as substrate after 90 mins | J Med Chem 61: 6468-6490 (2018) Article DOI: 10.1021/acs.jmedchem.7b00782 BindingDB Entry DOI: 10.7270/Q28S4SHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50457466 (CHEMBL4206158) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
Jadavpur University Curated by ChEMBL | Assay Description Inhibition of porcine kidney leucine aminopeptidase using LGG as substrate after 90 mins | J Med Chem 61: 6468-6490 (2018) Article DOI: 10.1021/acs.jmedchem.7b00782 BindingDB Entry DOI: 10.7270/Q28S4SHS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM23971 ((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.12E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534075 (CHEMBL4483393) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.65E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534075 (CHEMBL4483393) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.36E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 10 hrs measured every 6 mins by fluor... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM7460 (2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 3.43E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of pig kidney cytosolic Leucyl aminopeptidase | J Nat Prod 58: 823-829 (1995) Article DOI: 10.1021/np50120a001 BindingDB Entry DOI: 10.7270/Q2K937J6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM50157555 (2-(3,4-dihydroxyphenyl)-4H-chromen-4-one | 3',4'-d...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 3.51E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of pig kidney cytosolic Leucyl aminopeptidase | J Nat Prod 58: 823-829 (1995) Article DOI: 10.1021/np50120a001 BindingDB Entry DOI: 10.7270/Q2K937J6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase [33-68,L62W] (Sus scrofa (Pig)) | BDBM7459 (2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 4.96E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of pig kidney cytosolic Leucyl aminopeptidase | J Nat Prod 58: 823-829 (1995) Article DOI: 10.1021/np50120a001 BindingDB Entry DOI: 10.7270/Q2K937J6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534077 (CHEMBL4464704) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.36E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534070 (CHEMBL4454667) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.83E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534074 (CHEMBL4468968) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.93E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534069 (CHEMBL4473220) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.68E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534072 (CHEMBL4455383) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.11E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534078 (CHEMBL4557950) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.38E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534081 (CHEMBL4460083) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.63E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534071 (CHEMBL4563759) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.79E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534080 (CHEMBL4576374) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.09E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534073 (CHEMBL4537106) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.81E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534076 (CHEMBL4435767) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.05E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosol aminopeptidase (Sus scrofa) | BDBM50534079 (CHEMBL4456116) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.11E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Public Health-National Institute of Hygiene Curated by ChEMBL | Assay Description Inhibition of porcine kidney microsomal LAP using l-leucine-7-amido-4-methylcoumarin as substrate incubated for 60 mins measured every 3 mins by fluo... | Bioorg Med Chem 24: 5302-5314 (2016) Article DOI: 10.1016/j.bmc.2016.08.054 BindingDB Entry DOI: 10.7270/Q2NK3JHV | |||||||||||
More data for this Ligand-Target Pair |