Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314865 (CHEMBL4172616) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238185 (US9394303, 57) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | 130 | -9.39 | 670 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238190 (US9394303, 16) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 210 | -9.10 | 1.11E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238186 (US9394303, 58) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 250 | -9.00 | 1.28E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238181 (US9394303, 8) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 290 | -8.91 | 1.52E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314860 (CHEMBL4161200) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 340 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314864 (CHEMBL4172927) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314859 (CHEMBL4169123) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238192 (US9394303, 18) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 490 | -8.60 | 2.54E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314863 (CHEMBL4162253) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 490 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50315690 (CHEMBL4177447) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | Article PubMed | 560 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonism of carbachol action on nAChR of isolated frog rectus abdominus. | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314870 (CHEMBL4160019) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 740 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonist activity against Nicotinic acetylcholine receptor (nAChR) of isolated Frog rectus Abdominis Muscle | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238187 (US9394303, 59) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 820 | -8.30 | 4.27E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238196 (US9394303, 62) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 880 | -8.26 | 4.51E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238184 (US9394303, 56) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 900 | -8.24 | 4.68E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314874 (CHEMBL4176611) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314862 (CHEMBL4169534) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.08E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238191 (US9394303, 17) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.21E+3 | -8.07 | 6.30E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238195 (US9394303, 61) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.30E+3 | -8.02 | 6.76E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314861 (CHEMBL4177395) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238180 (US9394303, 7) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.40E+3 | -7.98 | 7.30E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238182 (US9394303, 9) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.40E+3 | -7.98 | 7.30E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50357753 (CHEMBL1916191) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington Curated by ChEMBL | Assay Description Displacement of BODIPY-Bak conjugated peptide from GST-tagged mouse wild type MCL1 expressed in Escherichia coli BL21 cells at 10 uM after 3 hrs by f... | Bioorg Med Chem Lett 21: 4951-5 (2011) Article DOI: 10.1016/j.bmcl.2011.06.134 BindingDB Entry DOI: 10.7270/Q2DB8287 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314855 (CHEMBL4176314) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.52E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238194 (US9394303, 60) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.53E+3 | -7.93 | 7.97E+3 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50357752 (CHEMBL1916190) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington Curated by ChEMBL | Assay Description Displacement of BODIPY-Bak conjugated peptide from GST-tagged mouse wild type MCL1 expressed in Escherichia coli BL21 cells at 10 uM after 3 hrs by f... | Bioorg Med Chem Lett 21: 4951-5 (2011) Article DOI: 10.1016/j.bmcl.2011.06.134 BindingDB Entry DOI: 10.7270/Q2DB8287 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50357756 (CHEMBL1916194) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington Curated by ChEMBL | Assay Description Displacement of BODIPY-Bak conjugated peptide from GST-tagged mouse wild type MCL1 expressed in Escherichia coli BL21 cells at 10 uM after 3 hrs by f... | Bioorg Med Chem Lett 21: 4951-5 (2011) Article DOI: 10.1016/j.bmcl.2011.06.134 BindingDB Entry DOI: 10.7270/Q2DB8287 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50357755 (CHEMBL1916193) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington Curated by ChEMBL | Assay Description Displacement of BODIPY-Bak conjugated peptide from GST-tagged mouse wild type MCL1 expressed in Escherichia coli BL21 cells at 10 uM after 3 hrs by f... | Bioorg Med Chem Lett 21: 4951-5 (2011) Article DOI: 10.1016/j.bmcl.2011.06.134 BindingDB Entry DOI: 10.7270/Q2DB8287 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238183 (US9394303, 10) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 2.06E+3 | -7.75 | 1.07E+4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50315693 (CHEMBL4166826) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 2.07E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238193 (US9394303, 55) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 2.09E+3 | -7.74 | 1.09E+4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50315549 (CHEMBL4175537) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 2.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonism of carbachol action on nAChR of isolated frog rectus abdominus. | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238189 (US9394303, 15) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 2.39E+3 | -7.66 | 1.24E+4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50119 (1-(3-chlorophenyl)-6-(2-furanyl)-3-methyl-4-pyrazo...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | US Patent | 2.64E+3 | -7.60 | 1.37E+4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238188 (US9394303, 14) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.32E+3 | -7.47 | 1.73E+4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238179 (US9394303, 6) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 3.54E+3 | -7.43 | 1.84E+4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314877 (CHEMBL4171691) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 3.55E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonism of carbachol action on nAChR of isolated frog rectus abdominus. | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314947 (CHEMBL4175134) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonism of carbachol action on nAChR of isolated frog rectus abdominus. | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM96413 (6-(2-furanyl)-3-methyl-1-phenyl-4-pyrazolo[3,4-b]p...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | US Patent | 4.25E+3 | -7.32 | 2.21E+4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314873 (CHEMBL4174087) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonist activity against Nicotinic acetylcholine receptor (nAChR) of isolated Frog rectus Abdominis Muscle | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314876 (CHEMBL4163814) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.74E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314866 (CHEMBL4161959) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314854 (CHEMBL4165700) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 5.92E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314875 (CHEMBL4168747) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Inhibition of FITC-Ahx-Bid-OH binding to mouse DN150/DC25 Mcl-1 after 2 hrs by fluorescent polarization assay | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314884 (CHEMBL4167271) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 6.83E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonism of carbachol action on nAChR of isolated frog rectus abdominus. | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50314869 (CHEMBL4167274) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 8.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonist activity against Nicotinic acetylcholine receptor (nAChR) of isolated Frog rectus Abdominis Muscle | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM21434 (N-Benylpiperazine derivative, 23j | N-[(4-{[(2R)-4...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington Curated by ChEMBL | Assay Description Displacement of BODIPY-Bak conjugated peptide from GST-tagged mouse wild type MCL1 expressed in Escherichia coli BL21 cells at 10 uM after 3 hrs by f... | Bioorg Med Chem Lett 21: 4951-5 (2011) Article DOI: 10.1016/j.bmcl.2011.06.134 BindingDB Entry DOI: 10.7270/Q2DB8287 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50357754 (CHEMBL1916192) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Washington Curated by ChEMBL | Assay Description Displacement of BODIPY-Bak conjugated peptide from GST-tagged mouse wild type MCL1 expressed in Escherichia coli BL21 cells at 10 uM after 3 hrs by f... | Bioorg Med Chem Lett 21: 4951-5 (2011) Article DOI: 10.1016/j.bmcl.2011.06.134 BindingDB Entry DOI: 10.7270/Q2DB8287 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM50315670 (CHEMBL4164915) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.37E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ Paris-Saclay Curated by ChEMBL | Assay Description Antagonism of carbachol action on nAChR of isolated frog rectus abdominus. | Eur J Med Chem 148: 26-38 (2018) Article DOI: 10.1016/j.ejmech.2018.01.100 BindingDB Entry DOI: 10.7270/Q2DF6TRW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 homolog (Mus musculus (Mouse)) | BDBM238177 (US9394303, 4) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | 1.46E+4 | -6.59 | 7.57E+4 | n/a | n/a | n/a | n/a | 7.4 | 25 |
THE REGENTS OF THE UNIVERSITY OF MICHIGAN US Patent | Assay Description Sensitive and quantitative FP-based binding assays were developed and optimized to determine the binding affinities of small-molecule inhibitors to t... | US Patent US9394303 (2016) BindingDB Entry DOI: 10.7270/Q2RJ4HCM | |||||||||||
More data for this Ligand-Target Pair |
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