Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362414 (CHEMBL1940537) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assay | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362412 (CHEMBL1940539) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assay | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362409 (CHEMBL1940543) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assay | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362412 (CHEMBL1940539) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by... | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362410 (CHEMBL1940542) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assay | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362415 (CHEMBL1940536) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assay | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50553728 (CHEMBL4757321) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1021/acs.jmedchem.1c01803 BindingDB Entry DOI: 10.7270/Q2KD22XQ | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50553728 (CHEMBL4757321) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assay | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127510 BindingDB Entry DOI: 10.7270/Q2RN3CHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362413 (CHEMBL1940538) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assay | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362413 (CHEMBL1940538) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 39 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by... | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362414 (CHEMBL1940537) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by... | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50553729 (CHEMBL4796786) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 53 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assay | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127510 BindingDB Entry DOI: 10.7270/Q2RN3CHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362409 (CHEMBL1940543) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by... | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50553730 (CHEMBL4779758) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assay | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127510 BindingDB Entry DOI: 10.7270/Q2RN3CHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50603458 (CHEMBL5196275) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 71 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.ejmech.2022.114149 BindingDB Entry DOI: 10.7270/Q2CN780J | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362411 (CHEMBL1940541) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 95 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assay | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425599 (CHEMBL2314291) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362415 (CHEMBL1940536) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 110 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by... | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50603462 (CHEMBL5198182) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 113 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.ejmech.2022.114149 BindingDB Entry DOI: 10.7270/Q2CN780J | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425598 (CHEMBL1972527) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425597 (CHEMBL2314320) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50401576 (CHEMBL2207117) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 160 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assay | Bioorg Med Chem Lett 22: 7135-41 (2012) Article DOI: 10.1016/j.bmcl.2012.09.074 BindingDB Entry DOI: 10.7270/Q2WS8VDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362410 (CHEMBL1940542) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 197 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by... | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50553719 (CHEMBL4744579) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 205 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assay | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127510 BindingDB Entry DOI: 10.7270/Q2RN3CHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50401572 (CHEMBL2207121) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assay | Bioorg Med Chem Lett 22: 7135-41 (2012) Article DOI: 10.1016/j.bmcl.2012.09.074 BindingDB Entry DOI: 10.7270/Q2WS8VDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425595 (CHEMBL2314323) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425596 (CHEMBL1981304) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50401577 (CHEMBL2207531) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assay | Bioorg Med Chem Lett 22: 7135-41 (2012) Article DOI: 10.1016/j.bmcl.2012.09.074 BindingDB Entry DOI: 10.7270/Q2WS8VDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425594 (CHEMBL1987422) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425593 (CHEMBL2314301) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425591 (CHEMBL2314300) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425592 (CHEMBL2314293) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425590 (CHEMBL1964671) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75901 (5-chloranyl-2-(3,5-dimethylphenyl)-4-(4-methoxyphe...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assay | Bioorg Med Chem Lett 22: 7135-41 (2012) Article DOI: 10.1016/j.bmcl.2012.09.074 BindingDB Entry DOI: 10.7270/Q2WS8VDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75938 (5-chloranyl-4-(4-methoxyphenoxy)-2-(4-propan-2-ylp...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assay | Bioorg Med Chem Lett 22: 7135-41 (2012) Article DOI: 10.1016/j.bmcl.2012.09.074 BindingDB Entry DOI: 10.7270/Q2WS8VDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75901 (5-chloranyl-2-(3,5-dimethylphenyl)-4-(4-methoxyphe...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75938 (5-chloranyl-4-(4-methoxyphenoxy)-2-(4-propan-2-ylp...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Molecular Screening Center Curated by PubChem BioAssay | Assay Description Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2GB22HQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75901 (5-chloranyl-2-(3,5-dimethylphenyl)-4-(4-methoxyphe...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 272 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Molecular Screening Center Curated by PubChem BioAssay | Assay Description Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2GB22HQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425589 (CHEMBL1969065) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75900 (5-chloranyl-4-(4-methoxyphenoxy)-2-(3-propan-2-ylp...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assay | Bioorg Med Chem Lett 22: 7135-41 (2012) Article DOI: 10.1016/j.bmcl.2012.09.074 BindingDB Entry DOI: 10.7270/Q2WS8VDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75900 (5-chloranyl-4-(4-methoxyphenoxy)-2-(3-propan-2-ylp...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 280 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Molecular Screening Center Curated by PubChem BioAssay | Assay Description Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2GB22HQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75901 (5-chloranyl-2-(3,5-dimethylphenyl)-4-(4-methoxyphe...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 281 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Molecular Screening Center Curated by PubChem BioAssay | Assay Description Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2XD1049 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50553720 (CHEMBL4754194) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 282 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human NPBWR1 assessed as inhibition of agonist-induced cAMP accumulation by cAMP assay | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127510 BindingDB Entry DOI: 10.7270/Q2RN3CHD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75946 (2-[3,5-bis(chloranyl)phenyl]-5-chloranyl-4-(4-meth...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 287 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Molecular Screening Center Curated by PubChem BioAssay | Assay Description Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2GB22HQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425588 (CHEMBL1965488) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 290 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75918 (5-chloranyl-4-(4-methoxyphenoxy)-2-(3-methyl-4-pro...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PCBioAssay | n/a | n/a | 299 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Molecular Screening Center Curated by PubChem BioAssay | Assay Description Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa... | PubChem Bioassay (2010) BindingDB Entry DOI: 10.7270/Q2GB22HQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM75918 (5-chloranyl-4-(4-methoxyphenoxy)-2-(3-methyl-4-pro...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in HEK293T cells co-expressing Galphaqi3 assessed as calcium release after 15 mins by FLIPR assay assay | Bioorg Med Chem Lett 22: 7135-41 (2012) Article DOI: 10.1016/j.bmcl.2012.09.074 BindingDB Entry DOI: 10.7270/Q2WS8VDC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50425587 (CHEMBL2314318) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
The Scripps Research Institute Curated by ChEMBL | Assay Description Antagonist activity against human NPBWR1 expressed in HEK293 cells co-expressing Gqi3 assessed as inhibition of agonist-induced response by FLIPR ass... | Bioorg Med Chem Lett 23: 614-9 (2013) Article DOI: 10.1016/j.bmcl.2012.12.030 BindingDB Entry DOI: 10.7270/Q20V8F30 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362416 (CHEMBL1940354) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 324 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Displacement of [125]-hNPW23 from human NPBWR1 expressed in CHO-K1 cells membrane by scintillation proximity assay | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptides B/W receptor type 1 (Homo sapiens (Human)) | BDBM50362411 (CHEMBL1940541) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 342 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Antagonist activity at human NPBWR1 expressed in CHO-K1 cells assessed as inhibition of hNPW23 and forskolin-stimulated cAMP production after 1 hr by... | Bioorg Med Chem Lett 22: 1014-8 (2012) Article DOI: 10.1016/j.bmcl.2011.11.126 BindingDB Entry DOI: 10.7270/Q2P84CB4 | |||||||||||
More data for this Ligand-Target Pair |
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