BindingDB PrimarySearch

Found 5 hits of ic50 for UniProtKB: P11167
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Solute carrier family 2, facilitated glucose transporter member 1 (Rattus norvegicus)	BDBM50250177 (((2R,3S,4S,5R,6R)-3,4,5,6-tetrahydroxytetrahydro-2...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	710	n/a	n/a	n/a	n/a	n/a	n/a
University of Kuopio Curated by ChEMBL					Assay Description Inhibition of GluT1-mediated [14C]D-glucose uptake in Wistar rat brain by perfusion technique				J Med Chem 52: 3348-53 (2009) Article DOI: 10.1021/jm8015409 BindingDB Entry DOI: 10.7270/Q2FQ9WHS
University of Kuopio Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 1 (Rattus norvegicus)	BDBM20877 (3-(1-benzofuran-5-yl)-1-(2-hydroxy-4-methyl-6-{[(2...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Mitsubishi Tanabe Pharma Corporation Curated by ChEMBL					Assay Description Inhibition of GLUT1-mediated [3H]2-deoxy-glucose uptake in rat L6 cells after 15 mins by liquid scintillation counting				J Med Chem 53: 6355-60 (2010) Article DOI: 10.1021/jm100332n BindingDB Entry DOI: 10.7270/Q2V69JSS
Mitsubishi Tanabe Pharma Corporation Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 1 (Rattus norvegicus)	BDBM50326284 (1-(beta-D-Glucopyranosyl)-4-methyl-3-(5-(4-fluorop...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
Mitsubishi Tanabe Pharma Corporation Curated by ChEMBL					Assay Description Inhibition of GLUT1-mediated [3H]2-deoxy-glucose uptake in rat L6 cells after 15 mins by liquid scintillation counting				J Med Chem 53: 6355-60 (2010) Article DOI: 10.1021/jm100332n BindingDB Entry DOI: 10.7270/Q2V69JSS
Mitsubishi Tanabe Pharma Corporation Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 1 (Rattus norvegicus)	BDBM50250141 (((2R,3S,4S,5R,6R)-3,4,5,6-tetrahydroxytetrahydro-2...) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	3.29E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Kuopio Curated by ChEMBL					Assay Description Inhibition of GluT1-mediated [14C]D-glucose uptake in Wistar rat brain by perfusion technique				J Med Chem 52: 3348-53 (2009) Article DOI: 10.1021/jm8015409 BindingDB Entry DOI: 10.7270/Q2FQ9WHS
University of Kuopio Curated by ChEMBL					More data for this Ligand-Target Pair
Solute carrier family 2, facilitated glucose transporter member 1 (Rattus norvegicus)	BDBM50277370 (CHEMBL4171968) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
Emory University Curated by ChEMBL					Assay Description Antagonist activity at rat C-terminal 6His/Myc-tagged GLUT1 assessed as reduction in 2-[3H]deoxyglucose uptake measured after 6 mins				Eur J Med Chem 139: 573-586 (2017) Article DOI: 10.1016/j.ejmech.2017.08.029 BindingDB Entry DOI: 10.7270/Q2NC63Q7
Emory University Curated by ChEMBL					More data for this Ligand-Target Pair