Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450899 (CHEMBL4214962) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 400 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450898 (CHEMBL4204476) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450897 (CHEMBL4202689) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.10E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450900 (CHEMBL4217485) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.40E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450901 (CHEMBL4211403) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as decrease in histone H3 citrulination incubated for 3 hrs in presence of ionomyc... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450897 (CHEMBL4202689) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.90E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450898 (CHEMBL4204476) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.50E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450900 (CHEMBL4217485) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.60E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450901 (CHEMBL4211403) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 8.30E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450899 (CHEMBL4214962) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 9.50E+3 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-arginine deiminase type-2 (Homo sapiens (Human)) | BDBM50450902 (CHEMBL4216140) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.06E+4 | n/a | n/a | n/a | n/a |
University of Massachusetts Medical School Curated by ChEMBL | Assay Description Binding affinity to human PAD2 expressed in HEK293T cells assessed as protein occupancy preincubated for 15 mins followed by ionomycin addition measu... | J Med Chem 60: 3198-3211 (2017) Article DOI: 10.1021/acs.jmedchem.7b00274 BindingDB Entry DOI: 10.7270/Q2SN0CJ1 | |||||||||||
More data for this Ligand-Target Pair |