Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467114 (CHEMBL4285682) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
LifeArc Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum protein kinase G | Bioorg Med Chem Lett 28: 3168-3173 (2018) Article DOI: 10.1016/j.bmcl.2018.08.028 BindingDB Entry DOI: 10.7270/Q21Z473B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467117 (CHEMBL4288816) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
LifeArc Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum protein kinase G | Bioorg Med Chem Lett 28: 3168-3173 (2018) Article DOI: 10.1016/j.bmcl.2018.08.028 BindingDB Entry DOI: 10.7270/Q21Z473B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530642 (CHEMBL4531058) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530642 (CHEMBL4531058) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.600 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467123 (CHEMBL4288103) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
LifeArc Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum protein kinase G | Bioorg Med Chem Lett 28: 3168-3173 (2018) Article DOI: 10.1016/j.bmcl.2018.08.028 BindingDB Entry DOI: 10.7270/Q21Z473B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467126 (CHEMBL4286880) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
LifeArc Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum protein kinase G | Bioorg Med Chem Lett 28: 3168-3173 (2018) Article DOI: 10.1016/j.bmcl.2018.08.028 BindingDB Entry DOI: 10.7270/Q21Z473B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467122 (CHEMBL4279865) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
LifeArc Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum protein kinase G | Bioorg Med Chem Lett 28: 3168-3173 (2018) Article DOI: 10.1016/j.bmcl.2018.08.028 BindingDB Entry DOI: 10.7270/Q21Z473B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530662 (CHEMBL4459320) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530662 (CHEMBL4459320) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530656 (CHEMBL4449947) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530653 (CHEMBL4469667) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530656 (CHEMBL4449947) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530663 (CHEMBL4532321) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530663 (CHEMBL4532321) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530649 (CHEMBL4451783) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530653 (CHEMBL4469667) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530649 (CHEMBL4451783) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530639 (CHEMBL4461276) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530639 (CHEMBL4461276) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467123 (CHEMBL4288103) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467123 (CHEMBL4288103) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467128 (CHEMBL4286841) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467128 (CHEMBL4286841) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50467128 (CHEMBL4286841) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
LifeArc Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum protein kinase G | Bioorg Med Chem Lett 28: 3168-3173 (2018) Article DOI: 10.1016/j.bmcl.2018.08.028 BindingDB Entry DOI: 10.7270/Q21Z473B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530660 (CHEMBL4455587) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530660 (CHEMBL4455587) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530661 (CHEMBL4593717) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530661 (CHEMBL4593717) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530652 (CHEMBL4572858) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50182362 (4-(7-((dimethylamino)methyl)-2-(4-fluorophenyl)H-i...) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
LifeArc Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum protein kinase G | Bioorg Med Chem Lett 28: 3168-3173 (2018) Article DOI: 10.1016/j.bmcl.2018.08.028 BindingDB Entry DOI: 10.7270/Q21Z473B | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530652 (CHEMBL4572858) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530647 (CHEMBL4585607) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530647 (CHEMBL4585607) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530646 (CHEMBL4531226) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530668 (CHEMBL4444451) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530668 (CHEMBL4444451) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530646 (CHEMBL4531226) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530651 (CHEMBL4566588) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530651 (CHEMBL4566588) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530640 (CHEMBL4546641) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530640 (CHEMBL4546641) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530637 (CHEMBL4591417) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530637 (CHEMBL4591417) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530650 (CHEMBL4459919) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.80 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530650 (CHEMBL4459919) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.80 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530654 (CHEMBL4446015) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530654 (CHEMBL4446015) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530666 (CHEMBL4446024) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50530666 (CHEMBL4446024) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum full length N-terminal His-tagged PKG expressed in Escherichia coli RosettaTM 2(DE3) pLysS cells using FAM-GRTGRR... | J Med Chem 62: 9217-9235 (2019) Article DOI: 10.1021/acs.jmedchem.9b01099 BindingDB Entry DOI: 10.7270/Q2X63RDP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cGMP-dependent protein kinase (Plasmodium falciparum) | BDBM50168171 (4-(2-(4-fluorophenyl)-5-(1-methylpiperidin-4-yl)-1...) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
LifeArc Curated by ChEMBL | Assay Description Inhibition of Plasmodium falciparum protein kinase G | Bioorg Med Chem Lett 28: 3168-3173 (2018) Article DOI: 10.1016/j.bmcl.2018.08.028 BindingDB Entry DOI: 10.7270/Q21Z473B | |||||||||||
More data for this Ligand-Target Pair |
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