Compile Data Set for Download or QSAR

Found 90 hits Enz. Inhib. hit(s) with all data for entry = 50047975   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM175970 (US10047103, 3 | US9605024, Example 3 | US9688695, ...) Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccccc3)cc(OC)cc2o1 Show InChI InChI=1S/C24H18N4O4S2/c1-29-16-8-19(31-12-15-13-33-22(25-15)14-6-4-3-5-7-14)17-10-21(32-20(17)9-16)18-11-28-23(26-18)34-24(27-28)30-2/h3-11,13H,12H2,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.00400	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 (unknown origin) assessed as inhibition of activating peptide-induced receptor activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM175970 (US10047103, 3 | US9605024, Example 3 | US9688695, ...) Show SMILES COc1nn2cc(nc2s1)-c1cc2c(OCc3csc(n3)-c3ccccc3)cc(OC)cc2o1 Show InChI InChI=1S/C24H18N4O4S2/c1-29-16-8-19(31-12-15-13-33-22(25-15)14-6-4-3-5-7-14)17-10-21(32-20(17)9-16)18-11-28-23(26-18)34-24(27-28)30-2/h3-11,13H,12H2,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	0.0230	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 (unknown origin) assessed as inhibition of gamma-thrombin-induced receptor activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199438 (CHEMBL3931873) Show SMILES COc1nn2cc(nc2s1)-c1cc2ccccc2o1 Show InChI InChI=1S/C13H9N3O2S/c1-17-13-15-16-7-9(14-12(16)19-13)11-6-8-4-2-3-5-10(8)18-11/h2-7H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.70	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 (unknown origin) assessed as inhibition of activating peptide-induced receptor activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199421 (CHEMBL3906197) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-2-4-8(5-3-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199421 (CHEMBL3906197) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-2-4-8(5-3-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	15	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199421 (CHEMBL3906197) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-2-4-8(5-3-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	16	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199420 (CHEMBL3933579) Show SMILES COc1nn2cc(nc2s1)-c1cc2cc(OC(F)(F)F)ccc2n1C Show InChI InChI=1S/C15H11F3N4O2S/c1-21-11-4-3-9(24-15(16,17)18)5-8(11)6-12(21)10-7-22-13(19-10)25-14(20-22)23-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	21	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199416 (CHEMBL3936444) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)(F)F)cc1 Show InChI InChI=1S/C12H8F3N3O2S/c1-19-11-17-18-6-9(16-10(18)21-11)7-2-4-8(5-3-7)20-12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	27	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199416 (CHEMBL3936444) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)(F)F)cc1 Show InChI InChI=1S/C12H8F3N3O2S/c1-19-11-17-18-6-9(16-10(18)21-11)7-2-4-8(5-3-7)20-12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	27	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199440 (CHEMBL3909608) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)c(Cl)c1 Show InChI InChI=1S/C11H7Cl2N3OS/c1-17-11-15-16-5-9(14-10(16)18-11)6-2-3-7(12)8(13)4-6/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199416 (CHEMBL3936444) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)(F)F)cc1 Show InChI InChI=1S/C12H8F3N3O2S/c1-19-11-17-18-6-9(16-10(18)21-11)7-2-4-8(5-3-7)20-12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199440 (CHEMBL3909608) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)c(Cl)c1 Show InChI InChI=1S/C11H7Cl2N3OS/c1-17-11-15-16-5-9(14-10(16)18-11)6-2-3-7(12)8(13)4-6/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	29	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199425 (CHEMBL3950308) Show SMILES COc1nn2cc(nc2s1)-c1cccc(c1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-3-2-4-8(5-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	36	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199425 (CHEMBL3950308) Show SMILES COc1nn2cc(nc2s1)-c1cccc(c1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-3-2-4-8(5-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	36	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199423 (CHEMBL3983476) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-2-4-8(12)5-3-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199423 (CHEMBL3983476) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-2-4-8(12)5-3-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199431 (CHEMBL3927486) Show SMILES COc1nn2cc(nc2s1)-c1cc(cc(c1)C(F)(F)F)C(F)(F)F Show InChI InChI=1S/C13H7F6N3OS/c1-23-11-21-22-5-9(20-10(22)24-11)6-2-7(12(14,15)16)4-8(3-6)13(17,18)19/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	52	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199431 (CHEMBL3927486) Show SMILES COc1nn2cc(nc2s1)-c1cc(cc(c1)C(F)(F)F)C(F)(F)F Show InChI InChI=1S/C13H7F6N3OS/c1-23-11-21-22-5-9(20-10(22)24-11)6-2-7(12(14,15)16)4-8(3-6)13(17,18)19/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	52	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199442 (CHEMBL3922644) Show SMILES COc1nn2cc(nc2s1)-c1ccc(C)cc1 Show InChI InChI=1S/C12H11N3OS/c1-8-3-5-9(6-4-8)10-7-15-11(13-10)17-12(14-15)16-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	57	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199442 (CHEMBL3922644) Show SMILES COc1nn2cc(nc2s1)-c1ccc(C)cc1 Show InChI InChI=1S/C12H11N3OS/c1-8-3-5-9(6-4-8)10-7-15-11(13-10)17-12(14-15)16-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	58	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199438 (CHEMBL3931873) Show SMILES COc1nn2cc(nc2s1)-c1cc2ccccc2o1 Show InChI InChI=1S/C13H9N3O2S/c1-17-13-15-16-7-9(14-12(16)19-13)11-6-8-4-2-3-5-10(8)18-11/h2-7H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	59	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 (unknown origin) assessed as inhibition of gamma-thrombin-induced receptor activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199433 (CHEMBL3902806) Show SMILES COc1nn2cc(nc2s1)-c1ccc(F)c(c1)C(F)(F)F Show InChI InChI=1S/C12H7F4N3OS/c1-20-11-18-19-5-9(17-10(19)21-11)6-2-3-8(13)7(4-6)12(14,15)16/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	69	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199433 (CHEMBL3902806) Show SMILES COc1nn2cc(nc2s1)-c1ccc(F)c(c1)C(F)(F)F Show InChI InChI=1S/C12H7F4N3OS/c1-20-11-18-19-5-9(17-10(19)21-11)6-2-3-8(13)7(4-6)12(14,15)16/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	69	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199428 (CHEMBL3890362) Show SMILES COc1nn2cc(nc2s1)-c1cccc(Cl)c1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-3-2-4-8(12)5-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	72	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199428 (CHEMBL3890362) Show SMILES COc1nn2cc(nc2s1)-c1cccc(Cl)c1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-3-2-4-8(12)5-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	73	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199418 (CHEMBL3973767) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)F)cc1 Show InChI InChI=1S/C12H9F2N3O2S/c1-18-12-16-17-6-9(15-11(17)20-12)7-2-4-8(5-3-7)19-10(13)14/h2-6,10H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	83	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199418 (CHEMBL3973767) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)F)cc1 Show InChI InChI=1S/C12H9F2N3O2S/c1-18-12-16-17-6-9(15-11(17)20-12)7-2-4-8(5-3-7)19-10(13)14/h2-6,10H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	83	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199437 (CHEMBL3912611) Show SMILES COc1nn2cc(nc2s1)-c1ccc(F)cc1F Show InChI InChI=1S/C11H7F2N3OS/c1-17-11-15-16-5-9(14-10(16)18-11)7-3-2-6(12)4-8(7)13/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	174	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199437 (CHEMBL3912611) Show SMILES COc1nn2cc(nc2s1)-c1ccc(F)cc1F Show InChI InChI=1S/C11H7F2N3OS/c1-17-11-15-16-5-9(14-10(16)18-11)7-3-2-6(12)4-8(7)13/h2-5H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	175	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199427 (CHEMBL3937549) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)[N+]([O-])=O Show InChI InChI=1S/C11H8N4O3S/c1-18-11-13-14-6-9(12-10(14)19-11)7-2-4-8(5-3-7)15(16)17/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	207	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199427 (CHEMBL3937549) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)[N+]([O-])=O Show InChI InChI=1S/C11H8N4O3S/c1-18-11-13-14-6-9(12-10(14)19-11)7-2-4-8(5-3-7)15(16)17/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	209	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199416 (CHEMBL3936444) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)(F)F)cc1 Show InChI InChI=1S/C12H8F3N3O2S/c1-19-11-17-18-6-9(16-10(18)21-11)7-2-4-8(5-3-7)20-12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	229	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199416 (CHEMBL3936444) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)(F)F)cc1 Show InChI InChI=1S/C12H8F3N3O2S/c1-19-11-17-18-6-9(16-10(18)21-11)7-2-4-8(5-3-7)20-12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	246	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199423 (CHEMBL3983476) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-2-4-8(12)5-3-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	286	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199421 (CHEMBL3906197) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-2-4-8(5-3-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	347	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199421 (CHEMBL3906197) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-2-4-8(5-3-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	348	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199416 (CHEMBL3936444) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC(F)(F)F)cc1 Show InChI InChI=1S/C12H8F3N3O2S/c1-19-11-17-18-6-9(16-10(18)21-11)7-2-4-8(5-3-7)20-12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	352	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199421 (CHEMBL3906197) Show SMILES COc1nn2cc(nc2s1)-c1ccc(cc1)C(F)(F)F Show InChI InChI=1S/C12H8F3N3OS/c1-19-11-17-18-6-9(16-10(18)20-11)7-2-4-8(5-3-7)12(13,14)15/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	398	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced P-selectin activation				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199424 (CHEMBL3946410) Show SMILES COc1nn2cc(nc2s1)-c1ccc(F)cc1 Show InChI InChI=1S/C11H8FN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-2-4-8(12)5-3-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	406	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199424 (CHEMBL3946410) Show SMILES COc1nn2cc(nc2s1)-c1ccc(F)cc1 Show InChI InChI=1S/C11H8FN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-2-4-8(12)5-3-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	407	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199435 (CHEMBL3894648) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1Cl Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-4-2-3-5-8(7)12/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	437	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199435 (CHEMBL3894648) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1Cl Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-4-2-3-5-8(7)12/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	437	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199439 (CHEMBL3955095) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1F Show InChI InChI=1S/C11H8FN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-4-2-3-5-8(7)12/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	525	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199439 (CHEMBL3955095) Show SMILES COc1nn2cc(nc2s1)-c1ccccc1F Show InChI InChI=1S/C11H8FN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-4-2-3-5-8(7)12/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	526	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199432 (CHEMBL3903596) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC)cc1 Show InChI InChI=1S/C12H11N3O2S/c1-16-9-5-3-8(4-6-9)10-7-15-11(13-10)18-12(14-15)17-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	589	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199432 (CHEMBL3903596) Show SMILES COc1nn2cc(nc2s1)-c1ccc(OC)cc1 Show InChI InChI=1S/C12H11N3O2S/c1-16-9-5-3-8(4-6-9)10-7-15-11(13-10)18-12(14-15)17-2/h3-7H,1-2H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	592	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair
Proteinase-activated receptor 4 (Homo sapiens (Human))	BDBM50199423 (CHEMBL3983476) Show SMILES COc1nn2cc(nc2s1)-c1ccc(Cl)cc1 Show InChI InChI=1S/C11H8ClN3OS/c1-16-11-14-15-6-9(13-10(15)17-11)7-2-4-8(12)5-3-7/h2-6H,1H3	UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	617	n/a	n/a	n/a	n/a	n/a	n/a
Vanderbilt University Medical Center Curated by ChEMBL					Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow...				Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD
					More data for this Ligand-Target Pair

Displayed 1 to 50 (of 90 total )  |  Next  |  Last  >>

Jump to: