Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Solute carrier family 22 member 2 (RAT) | BDBM50420215 (CHEMBL339858) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Heidelberg Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Dopamine uptake in OCT2-expressing HEK293 cells | J Biol Chem 273: 30915-20 (1998) BindingDB Entry DOI: 10.7270/Q2V40WGS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 2 (RAT) | BDBM50420215 (CHEMBL339858) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Heidelberg Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Adrenaline uptake in OCT2-expressing HEK293 cells | J Biol Chem 273: 30915-20 (1998) BindingDB Entry DOI: 10.7270/Q2V40WGS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 2 (RAT) | BDBM50420215 (CHEMBL339858) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Heidelberg Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Noradrenaline uptake in OCT2-expressing HEK293 cells | J Biol Chem 273: 30915-20 (1998) BindingDB Entry DOI: 10.7270/Q2V40WGS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 2 (RAT) | BDBM50420215 (CHEMBL339858) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Heidelberg Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Serotonin uptake in OCT2-expressing HEK293 cells | J Biol Chem 273: 30915-20 (1998) BindingDB Entry DOI: 10.7270/Q2V40WGS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 2 (RAT) | BDBM50170653 ((11beta)-11,21-dihydroxypregn-4-ene-3,20-dione | 1...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Heidelberg Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Dopamine uptake in OCT2-expressing HEK293 cells | J Biol Chem 273: 30915-20 (1998) BindingDB Entry DOI: 10.7270/Q2V40WGS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 2 (RAT) | BDBM50170653 ((11beta)-11,21-dihydroxypregn-4-ene-3,20-dione | 1...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Heidelberg Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Adrenaline uptake in OCT2-expressing HEK293 cells | J Biol Chem 273: 30915-20 (1998) BindingDB Entry DOI: 10.7270/Q2V40WGS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 2 (RAT) | BDBM50170653 ((11beta)-11,21-dihydroxypregn-4-ene-3,20-dione | 1...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 460 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Heidelberg Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Noradrenaline uptake in OCT2-expressing HEK293 cells | J Biol Chem 273: 30915-20 (1998) BindingDB Entry DOI: 10.7270/Q2V40WGS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 2 (RAT) | BDBM50170653 ((11beta)-11,21-dihydroxypregn-4-ene-3,20-dione | 1...) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 605 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Heidelberg Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of Serotonin uptake in OCT2-expressing HEK293 cells | J Biol Chem 273: 30915-20 (1998) BindingDB Entry DOI: 10.7270/Q2V40WGS | |||||||||||
More data for this Ligand-Target Pair |